SCHEMBL8764291

SCHEMBL8764291

Nc1onc(C(F)(F)C(F)(F)F)c1-c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.53
TDO2 P48775 1/20 0.53
MLYCD O95822 13/20 0.52
PTGS1 P23219 1/20 0.43
POLB P06746 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.38
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
NOTUM Q6P988 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8764932 0.86 MLYCD (0.63) BRD4TDO2MLYCDPTGS1POLB
SCHEMBL8765096 0.73 L3MBTL1 (0.45) BRD4TDO2MLYCDPTGS1POLB
SCHEMBL27744909 0.71 MLYCD (0.61) BRD4TDO2MLYCD
SCHEMBL10502800 0.71 MLYCD (0.66) BRD4TDO2MLYCD
SCHEMBL10503952 0.70 MLYCD (0.64) BRD4TDO2MLYCDPTGS1NOTUM
SCHEMBL544899 0.69 BRD4 (1.00) BRD4TDO2MLYCDPTGS1NOTUM
SCHEMBL4420017 0.69 MLYCD (1.00) MLYCDESR1ESR2
SCHEMBL4874434 0.69 MLYCD (1.00) MLYCD
SCHEMBL8765219 0.67 MLYCD (0.35) BRD4MLYCD
SCHEMBL10505666 0.67 MLYCD (0.59) MLYCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4797492-A INTERMEDIATES FOR BACTERICIDES; HERBICIDES OR FUNGICIDES SHIONOGI & CO., LTD. (JP) 1989-01-10 US claimed
EP-0220947-A2 Polyfluoroalkylisoxazolylamines, their preparation and use SHIONOGI & CO., LTD. (JP) 1987-05-06 EP claimed
EP-0375670-B1 Process for preparing 3-polyfluoroalkylisoxazolylamines SHIONOGI & CO (JP) 1997-08-06 EP disclosed
EP-0220947-B1 Polyfluoroalkylisoxazolylamines, their preparation and use SHIONOGI & CO (JP) 1994-06-15 EP disclosed
EP-0375670-A2 Process for preparing 3-polyfluoroalkylisoxazolylamines SHIONOGI & CO., LTD. (JP) 1990-06-27 EP disclosed
US-4797492-A INTERMEDIATES FOR BACTERICIDES; HERBICIDES OR FUNGICIDES SHIONOGI & CO., LTD. (JP) 1989-01-10 US disclosed
EP-0220947-A2 Polyfluoroalkylisoxazolylamines, their preparation and use SHIONOGI & CO., LTD. (JP) 1987-05-06 EP disclosed