SCHEMBL8764932

SCHEMBL8764932

Nc1onc(C(F)(F)F)c1-c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 7/20 0.63
BRD4 O60885 3/20 0.56
TDO2 P48775 2/20 0.56
POLB P06746 1/20 0.49
PTGS1 P23219 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
ENPP1 P22413 1/20 0.40
NOTUM Q6P988 1/20 0.38
BRD2 P25440 1/20 0.38
PTGS2 P35354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8764291 0.86 BRD4 (0.53) MLYCDBRD4TDO2POLBPTGS1
SCHEMBL10502800 0.84 MLYCD (0.66) MLYCDBRD4TDO2ENPP1PTGS2
SCHEMBL10503592 0.83 MLYCD (0.64) MLYCDBRD4TDO2ENPP1
SCHEMBL10503952 0.83 MLYCD (0.64) MLYCDBRD4TDO2PTGS1NOTUM
SCHEMBL10505666 0.79 MLYCD (0.59) MLYCDENPP1PTGS2
SCHEMBL9674379 0.79 PTGS1 (0.46) MLYCDBRD4TDO2POLBPTGS1
SCHEMBL4874434 0.78 MLYCD (1.00) MLYCD
SCHEMBL8764336 0.75 TDO2 (0.46) MLYCDBRD4TDO2POLBPTGS1
SCHEMBL10502923 0.72 MLYCD (0.52) MLYCDBRD4
SCHEMBL10731646 0.72 MLYCD (0.52) MLYCDBRD4POLBPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4797492-A INTERMEDIATES FOR BACTERICIDES; HERBICIDES OR FUNGICIDES SHIONOGI & CO., LTD. (JP) 1989-01-10 US claimed
EP-0220947-A2 Polyfluoroalkylisoxazolylamines, their preparation and use SHIONOGI & CO., LTD. (JP) 1987-05-06 EP claimed
EP-0375670-B1 Process for preparing 3-polyfluoroalkylisoxazolylamines SHIONOGI & CO (JP) 1997-08-06 EP disclosed
EP-0220947-B1 Polyfluoroalkylisoxazolylamines, their preparation and use SHIONOGI & CO (JP) 1994-06-15 EP disclosed
EP-0271975-B1 3-PERFLUOROALKYL-ISOXAZOL-5-YL-OXYCARBOXYLIC ACID DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1992-06-24 EP disclosed
EP-0375670-A2 Process for preparing 3-polyfluoroalkylisoxazolylamines SHIONOGI & CO., LTD. (JP) 1990-06-27 EP disclosed
US-4888044-A PREEMERGENCE HERBICIDES SHIONOGI & CO., LTD. (JP) 1989-12-19 US disclosed
US-4797492-A INTERMEDIATES FOR BACTERICIDES; HERBICIDES OR FUNGICIDES SHIONOGI & CO., LTD. (JP) 1989-01-10 US disclosed
EP-0271975-A1 3-Perfluoroalkyl-isoxazol-5-yl-oxycarboxylic acid derivatives, processes for their preparation and their use as herbicides SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1988-06-22 EP disclosed
EP-0220947-A2 Polyfluoroalkylisoxazolylamines, their preparation and use SHIONOGI & CO., LTD. (JP) 1987-05-06 EP disclosed