SCHEMBL27745447

SCHEMBL27745447

NC(=O)c1nn(-c2ccc(F)cc2Cl)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
NR3C2 P08235 1/20 0.39
PTPN11 Q06124 2/20 0.39
PARP1 P09874 2/20 0.39
GRM2 Q14416 1/20 0.37
P2RX7 Q99572 2/20 0.36
MARS1 P56192 1/20 0.36
CAPN1 P07384 1/20 0.35
GRIN2B Q13224 3/20 0.35
GRM5 P41594 1/20 0.35
ALOX15 P16050 2/20 0.34
NOTUM Q6P988 1/20 0.34
GRIN1 Q05586 1/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
CASP6 P55212 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4636950 0.90 ALDH1A1 (0.40) ALDH1A1NR3C2PTPN11PARP1GRM2
SCHEMBL20022423 0.74 HDAC9 (0.41) ALDH1A1NR3C2PARP1GRIN2BGRIN1
SCHEMBL3946970 0.73 ALDH1A1 (0.52) ALDH1A1NOTUM
SCHEMBL30108354 0.73 ALDH1A1 (0.52) ALDH1A1NOTUM
SCHEMBL30582191 0.73 GRM2 (0.41) ALDH1A1NR3C2GRM2P2RX7MARS1
SCHEMBL6506908 0.73 ITK (0.42) ALDH1A1NR3C2PARP1MEN1KMT2A
SCHEMBL6506387 0.72 ITK (0.41) ALDH1A1NR3C2MEN1KMT2A
SCHEMBL167526 0.72 AURKA (0.42) ALDH1A1P2RX7MARS1GRM5MEN1
SCHEMBL168945 0.72 AURKA (0.42) ALDH1A1P2RX7GRM5
SCHEMBL27724732 0.71 MARS1 (0.46) ALDH1A1NR3C2GRM2MARS1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101331118-A Pyrazoles useful in the treatment of inflammation BIOLIPOX AB (SE) 2008-12-24 CN disclosed