SCHEMBL27746212

SCHEMBL27746212

Nc1cccc2c1CC(N)C(=O)N2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.37
BRD4 O60885 2/20 0.36
TNF P01375 2/20 0.36
IL1B P01584 2/20 0.36
IKZF1 Q13422 2/20 0.36
DDB1 Q16531 2/20 0.36
CRBN Q96SW2 2/20 0.36
IKZF3 Q9UKT9 2/20 0.36
AADAT Q8N5Z0 3/20 0.33
CREBBP Q92793 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
BRPF1 P55201 1/20 0.33
HTR5A P47898 4/20 0.33
GSK3B P49841 1/20 0.33
IDO1 P14902 1/20 0.33
HTR1A P08908 1/20 0.33
HTR1D P28221 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29073375 0.81 CDK5 (0.38) BRD4AADATCREBBPKDM4EALDH1A1
SCHEMBL4067227 0.81 AADAT (0.49) BRD4DDB1CRBNAADATCREBBP
SCHEMBL1450613 0.81 PARP1 (0.36) PARP1BRD4TNFIL1BIKZF1
SCHEMBL13725343 0.81 AADAT (0.49) PARP1BRD4DDB1CRBNAADAT
Hydrochloric Acid SCHEMBL25331216 0.80 CDK5 (0.37) BRD4AADATCREBBPKDM4EALDH1A1
Hydrochloric Acid SCHEMBL30576552 0.80 CDK5 (0.37) BRD4AADATCREBBPKDM4EALDH1A1
Hydrochloric Acid SCHEMBL4894658 0.80 AADAT (0.48) PARP1BRD4DDB1CRBNAADAT
SCHEMBL4795933 0.78 AADAT (0.52) BRD4AADATCREBBPALDH1A1MAPT
SCHEMBL3593980 0.78 HTR5A (0.35) PARP1BRD4TNFIL1BIKZF1
SCHEMBL3591908 0.78 CREBBP (0.38) PARP1BRD4TNFIL1BIKZF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101489989-A Pentadiene amide derivative KYOWA HAKKO KIRIN CO LTD (JP) 2009-07-22 CN disclosed