SCHEMBL27763561

SCHEMBL27763561

CC(=O)Oc1nc(N[C@H](CO)Cc2ccccc2)c2nc[nH]c2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 1/20 0.40
CX3CR1 P49238 1/20 0.40
MME P08473 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
CDK1 P06493 2/20 0.39
CDK5 Q00535 2/20 0.39
ROCK2 O75116 3/20 0.39
ROCK1 Q13464 3/20 0.39
CYP3A4 P08684 1/20 0.38
MAPK1 P28482 1/20 0.38
JAK3 P52333 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
CCNE2 O96020 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
AURKA O14965 2/20 0.37
RPS6KB1 P23443 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1412351 0.82 KDM4E (0.40) MMEKDM4EMEN1MAPTKMT2A
SCHEMBL27763566 0.82 KDM4E (0.43) MMEKDM4EMEN1MAPTKMT2A
SCHEMBL27763565 0.82 KDM4E (0.43) MMEKDM4EMEN1MAPTKMT2A
SCHEMBL27763562 0.80 KDM4E (0.42) MMEKDM4EMEN1MAPTKMT2A
SCHEMBL27532522 0.77 ADORA2A (0.35) KMT2AROCK2ROCK1MAPK1
SCHEMBL7658491 0.72 KDM4E (0.44) MMEKDM4EMEN1MAPTKMT2A
SCHEMBL7085340 0.70 ADORA2A (0.47) MMEKDM4EMEN1MAPTKMT2A
SCHEMBL27564857 0.70 ADORA2A (0.47) MMEKDM4EMEN1MAPTKMT2A
Hydrochloric Acid SCHEMBL7088885 0.70 ADORA2A (0.47) MMEKDM4EMEN1MAPTKMT2A
SCHEMBL7088146 0.69 NPR3 (0.42) MMEMEN1MAPTKMT2ACDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101437829-B Bisadenosine compounds as adenosine A2A receptor agonists NOVARTIS AG 2012-03-21 CN disclosed
CN-101437829-A Bisadenosine compounds as adenosine A2A receptor agonists NOVARTIS AG (CH) 2009-05-20 CN disclosed