SCHEMBL4162283

SCHEMBL4162283

CCCS(=O)(=O)c1ccc(-c2cccc(-c3nc4c(C(F)(F)F)cccc4cc3C)c2Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 12/20 0.41
NR1H3 Q13133 8/20 0.41
CYP3A4 P08684 4/20 0.38
CYP2C9 P11712 4/20 0.38
CYP1A2 P05177 3/20 0.38
CYP2C19 P33261 3/20 0.38
CYP2D6 P10635 2/20 0.37
RORC P51449 2/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
HSD11B1 P28845 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4166161 0.93 NR1H2 (0.46) NR1H2NR1H3CYP3A4CYP2C9CYP1A2
SCHEMBL4167137 0.87 NR1H2 (0.46) NR1H2NR1H3
SCHEMBL4162285 0.81 NR1H2 (0.44) NR1H2NR1H3CYP3A4CYP2C9CYP1A2
SCHEMBL4165443 0.76 NR1H2 (0.44) NR1H2NR1H3CYP3A4CYP2C9CYP1A2
SCHEMBL27765403 0.75 NR1H2 (0.40) NR1H2NR1H3CYP3A4CYP2C9CYP1A2
SCHEMBL27765402 0.75 NR1H2 (0.40) NR1H2NR1H3RORCHSD11B1
SCHEMBL4166168 0.74 NR1H2 (0.48) NR1H2NR1H3RORC
SCHEMBL27786940 0.71 NR1H2 (0.42) NR1H2NR1H3
SCHEMBL4165449 0.71 NR1H2 (0.44) NR1H2NR1H3
SCHEMBL28780848 0.71 NR1H2 (0.39) NR1H2NR1H3HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed