SCHEMBL27766089

SCHEMBL27766089

CCN1CCNCC1.Fc1cccc(F)c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.51
SLC6A2 P23975 9/20 0.46
SLC6A4 P31645 7/20 0.45
SLC6A3 Q01959 3/20 0.45
KCNH2 Q12809 2/20 0.45
HTR6 P50406 2/20 0.43
HTR1A P08908 4/20 0.43
SIGMAR1 Q99720 1/20 0.42
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
CHRM3 P20309 1/20 0.41
HTR7 P34969 2/20 0.41
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluorobenzene SCHEMBL27488633 0.87 SIGMAR1 (0.52) KDM4ESLC6A2SLC6A4SIGMAR1HTR7
Tert-Butyl Formate SCHEMBL28022652 0.85 KDM4E (0.40) KDM4ESLC6A2SLC6A4SLC6A3KCNH2
Methylpiperazine SCHEMBL28021853 0.79 HTR1A (0.45) SLC6A2SLC6A4SLC6A3KCNH2HTR6
Methylpiperazine SCHEMBL28021851 0.78 HTR1A (0.44) SLC6A2SLC6A4SLC6A3KCNH2HTR6
SCHEMBL29566534 0.77 ALDH1A1 (0.70) KDM4ESIGMAR1CHRM3ALDH1A1SMN1; SMN2
SCHEMBL608181 0.77 ALDH1A1 (0.70) KDM4ESIGMAR1CHRM3ALDH1A1SMN1; SMN2
SCHEMBL1307906 0.77 HRH3 (0.46) SIGMAR1ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL2924548 0.76 ALDH1A1 (0.68) KDM4ESIGMAR1CHRM3ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL7426019 0.76 ALDH1A1 (0.68) KDM4ESIGMAR1CHRM3ALDH1A1SMN1; SMN2
SCHEMBL5943 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102838546-B Pyrazole derivatives as modulators of 5-ht2a serotonin receptor useful for treatment of disorders related thereto ARENA PHARM INC 2015-07-15 CN disclosed
CN-102838546-A Pyrazole derivatives as modulators of 5-ht2a serotonin receptor useful for treatment of disorders related thereto ARENA PHARM INC 2012-12-26 CN disclosed
CN-101611013-B As 5-HT2APyrazole derivatives of serotonin receptor modulators for the treatment of disorders related thereto ARENA PHARM INC 2012-09-05 CN disclosed
CN-101611013-A As 5-HT2APyrazole derivatives of serotonin receptor modulators for the treatment of disorders related thereto ARENA PHARM INC (US) 2009-12-23 CN disclosed