SCHEMBL27768129

SCHEMBL27768129

CC(=O)OCc1nc(C(=O)O)c(-c2ccccc2)s1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.55
CYP2C19 P33261 3/20 0.55
ALDH1A1 P00352 3/20 0.49
ALOX5 P09917 1/20 0.45
KDM4E B2RXH2 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HSD17B10 Q99714 2/20 0.44
HPGD P15428 1/20 0.44
GAA P10253 1/20 0.41
PPARD Q03181 4/20 0.39
CYP2C9 P11712 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
MAPK1 P28482 1/20 0.37
CASP1 P29466 1/20 0.37
PIN1 Q13526 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3316068 0.87 CYP1A2 (0.50) CYP1A2CYP2C19ALDH1A1KDM4ESMN1; SMN2
SCHEMBL27789562 0.79 KDM4E (0.47) CYP1A2CYP2C19ALDH1A1ALOX5KDM4E
SCHEMBL27789654 0.78 KDM4E (0.44) CYP1A2CYP2C19ALDH1A1ALOX5KDM4E
SCHEMBL13398494 0.78 KDM4E (0.46) CYP1A2CYP2C19ALDH1A1ALOX5KDM4E
SCHEMBL14705607 0.74 PTGS2 (0.39) ALDH1A1ALOX5KDM4ESMN1; SMN2HSD17B10
SCHEMBL80459 0.72 ALOX5 (0.61) CYP1A2CYP2C19ALDH1A1ALOX5KDM4E
SCHEMBL4328431 0.72 KDM4A (0.44) ALDH1A1KDM4ESMN1; SMN2HSD17B10HPGD
SCHEMBL13398512 0.72 KDM4E (0.52) CYP1A2CYP2C19ALDH1A1ALOX5KDM4E
SCHEMBL14705610 0.71 MAPK14 (0.39) CYP1A2ALDH1A1ALOX5HSD17B10CYP2C9
SCHEMBL3314567 0.71 TRPM8 (0.53) CYP1A2CYP2C19ALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101605784-B Aza-bridged-ring compound ASTELLAS PHARMA INC JP 2013-04-10 CN disclosed
CN-101605784-A Aza-bridged-ring compound ASTELLAS PHARMA INC (JP) 2009-12-16 CN disclosed