SCHEMBL27768402

SCHEMBL27768402

O=CNc1ccc2nccnc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 9/20 0.50
ALDH1A1 P00352 8/20 0.50
KDM4E B2RXH2 7/20 0.50
MAPT P10636 7/20 0.50
SMN1; SMN2 Q16637 5/20 0.50
ADRA2A P08913 2/20 0.47
ADRA2C P18825 2/20 0.47
NPC1 O15118 8/20 0.46
RAB9A P51151 8/20 0.46
HPGD P15428 3/20 0.46
TP53 P04637 3/20 0.46
GAA P10253 3/20 0.46
CASP1 P29466 2/20 0.46
CASP7 P55210 2/20 0.46
HSD17B10 Q99714 2/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
NFKB1 P19838 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19597819 0.81 MAPT (0.43) KMT2AALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL27840250 0.81 KMT2A (0.47) KMT2AALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL10133307 0.78 NPC1 (0.61) KMT2AALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL18789747 0.78 MEN1 (0.50) KMT2AALDH1A1MAPTNPC1CASP1
SCHEMBL27805824 0.78 ALDH1A1 (0.39) KMT2AALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL28067551 0.77 ALDH1A1 (0.38) KMT2AALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL28173261 0.77 MEN1 (0.49) KMT2AALDH1A1MAPTNPC1CASP1
SCHEMBL28152084 0.77 NPC1 (0.59) KMT2AALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL6203397 0.75 NR4A2 (0.51) KMT2AMAPTMEN1
SCHEMBL6579243 0.74 MAPT (0.45) KMT2AALDH1A1MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107108534-A Probes for Imaging Huntingtin CHDI基金会股份有限公司 2017-08-29 CN claimed
CN-107001345-A Hete rocyclic derivatives and application thereof 株式会社C&C新药研究所 2017-08-01 CN claimed
CN-101616919-B Poly (ADP ribose) polymerase inhibitors ABBOTT LAB 2012-10-10 CN claimed
CN-104788430-B The treatment method of pyrazole derivatives calcium release activation calcium channel modulators and non-small cell lung cancer 理森制药股份公司 2019-10-22 CN disclosed
CN-106458934-B Quinoxaline compounds and application thereof 米伦纽姆医药公司 2019-08-16 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed
CN-109310690-A Isoquinolin -3- base benzamide type and its preparation and its purposes 萨穆梅德有限公司 2019-02-05 CN disclosed
CN-108794411-A Certain chemical entities, composition and method 润新生物公司 2018-11-13 CN disclosed
CN-104080455-B Certain chemical entities, compositions, and methods 润新生物公司 2018-07-31 CN disclosed
CN-107245056-A Chemical entities, composition and method 润新生物公司 2017-10-13 CN disclosed
CN-107108534-A Probes for Imaging Huntingtin CHDI基金会股份有限公司 2017-08-29 CN disclosed
CN-107001345-A Hete rocyclic derivatives and application thereof 株式会社C&C新药研究所 2017-08-01 CN disclosed
CN-104053442-B Certain chemical entities, compositions, and methods 润新生物公司 2017-06-23 CN disclosed
CN-106458934-A Quinoxaline compounds and uses thereof 米伦纽姆医药公司 2017-02-22 CN disclosed
CN-101616919-B Poly (ADP ribose) polymerase inhibitors ABBOTT LAB 2012-10-10 CN disclosed
CN-102036561-A Protein kinase modulators CYLENE PHARMACEUTICALS INC 2011-04-27 CN disclosed
CN-101616919-A Poly (ADP ribose) polymerase inhibitors ABBOTT LAB 2009-12-30 CN disclosed