SCHEMBL27768408

SCHEMBL27768408

CC(=O)Oc1c(C)n(Cc2nc3ccccc3s2)c2cc(Cl)ccc12

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 3/20 0.52
AKR1B1 P15121 9/20 0.48
CYP1A2 P05177 1/20 0.45
CYP2C19 P33261 1/20 0.45
KLKB1 P03952 1/20 0.42
KLK1 P06870 1/20 0.42
P2RX7 Q99572 1/20 0.41
EPHX2 P34913 2/20 0.41
ALOX5 P09917 2/20 0.41
ALOX5AP P20292 1/20 0.41
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27789966 0.92 PTGDR2 (0.56) PTGDR2AKR1B1CYP1A2CYP2C19KLKB1
SCHEMBL27905712 0.85 PTGDR2 (0.49) PTGDR2AKR1B1CYP1A2CYP2C19KLKB1
SCHEMBL4778730 0.85 PTGDR2 (0.56) PTGDR2AKR1B1CYP1A2CYP2C19KLKB1
SCHEMBL27790170 0.84 PTGDR2 (0.50) PTGDR2AKR1B1CYP1A2CYP2C19KLKB1
SCHEMBL4777221 0.83 PTGDR2 (0.70) PTGDR2AKR1B1CYP1A2CYP2C19KLKB1
SCHEMBL2002085 0.82 PTGDR2 (0.70) PTGDR2AKR1B1ALOX5
SCHEMBL27768505 0.81 PTGDR2 (0.53) PTGDR2AKR1B1CYP1A2CYP2C19KLKB1
SCHEMBL27768501 0.79 PTGDR2 (0.56) PTGDR2AKR1B1CYP1A2CYP2C19KLKB1
SCHEMBL2001831 0.76 PTGDR2 (0.79) PTGDR2AKR1B1CYP1A2CYP2C19ALOX5
SCHEMBL4565555 0.74 PTGDR2 (0.66) PTGDR2AKR1B1CYP1A2CYP2C19ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102850324-A Indole compounds MICROBIA INC 2013-01-02 CN disclosed
CN-101563337-A Indole compounds MICROBIA INC (US) 2009-10-21 CN disclosed