SCHEMBL4777221

SCHEMBL4777221

CC(=O)Oc1c(C)n(Cc2nc3ccccc3s2)c2ccc(F)cc12

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 5/20 0.70
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
P2RX7 Q99572 1/20 0.46
KLKB1 P03952 1/20 0.42
KLK1 P06870 1/20 0.42
MAPT P10636 5/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
AKR1B1 P15121 4/20 0.41
PTGIR P43119 1/20 0.41
PTGDR Q13258 1/20 0.41
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
GAA P10253 1/20 0.40
ALDH1A1 P00352 3/20 0.40
USP2 O75604 1/20 0.40
TSHR P16473 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27789966 0.89 PTGDR2 (0.56) PTGDR2CYP1A2CYP2C19P2RX7KLKB1
SCHEMBL4778730 0.89 PTGDR2 (0.56) PTGDR2CYP1A2CYP2C19P2RX7KLKB1
SCHEMBL27768501 0.87 PTGDR2 (0.56) PTGDR2CYP1A2CYP2C19P2RX7KLKB1
SCHEMBL27768505 0.86 PTGDR2 (0.53) PTGDR2CYP1A2CYP2C19P2RX7KLKB1
SCHEMBL2010037 0.83 PTGDR2 (0.72) PTGDR2CYP1A2CYP2C19P2RX7KLKB1
SCHEMBL27768408 0.83 PTGDR2 (0.52) PTGDR2CYP1A2CYP2C19P2RX7KLKB1
SCHEMBL27790170 0.83 PTGDR2 (0.50) PTGDR2CYP1A2CYP2C19P2RX7KLKB1
SCHEMBL2005637 0.82 PTGDR2 (1.00) PTGDR2CYP1A2CYP2C19P2RX7KDM4E
SCHEMBL27905712 0.82 PTGDR2 (0.49) PTGDR2CYP1A2CYP2C19P2RX7KLKB1
SCHEMBL16558821 0.81 PTGDR2 (0.76) PTGDR2P2RX7KLKB1KLK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1931632-A2 USEFUL INDOLE COMPOUNDS Microbia Inc. (US) 2008-06-18 EP disclosed
WO-2007022501-A2 USEFUL INDOLE COMPOUNDS MICROBIA, INC. (US) 2007-02-22 WO disclosed