SCHEMBL27768501

SCHEMBL27768501

CC(=O)Oc1c(C)n(Cc2nc3ccccc3s2)c2ccc(OC(F)(F)F)cc12

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.56
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
AKR1B1 P15121 5/20 0.41
ALOX5AP P20292 4/20 0.40
ALOX5 P09917 1/20 0.40
MAPT P10636 2/20 0.39
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
KLKB1 P03952 1/20 0.39
KLK1 P06870 1/20 0.39
DYRK1A Q13627 1/20 0.39
ELANE P08246 1/20 0.39
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
F2RL3 Q96RI0 1/20 0.38
P2RX7 Q99572 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4777221 0.87 PTGDR2 (0.70) PTGDR2CYP1A2CYP2C19AKR1B1MAPT
SCHEMBL2003155 0.85 PTGDR2 (0.75) PTGDR2CYP1A2CYP2C19AKR1B1MAPT
SCHEMBL27789966 0.84 PTGDR2 (0.56) PTGDR2CYP1A2CYP2C19AKR1B1ALOX5AP
SCHEMBL27768505 0.83 PTGDR2 (0.53) PTGDR2CYP1A2CYP2C19AKR1B1MAPT
SCHEMBL4778730 0.83 PTGDR2 (0.56) PTGDR2CYP1A2CYP2C19AKR1B1MAPT
SCHEMBL27790170 0.82 PTGDR2 (0.50) PTGDR2CYP1A2CYP2C19AKR1B1ALOX5AP
SCHEMBL27768408 0.79 PTGDR2 (0.52) PTGDR2CYP1A2CYP2C19AKR1B1ALOX5AP
SCHEMBL27768704 0.78 PPARG (0.54) CYP1A2CYP2C19ALOX5CYP2D6CYP2C9
SCHEMBL27905712 0.78 PTGDR2 (0.49) PTGDR2CYP1A2CYP2C19AKR1B1ALOX5
SCHEMBL27889074 0.75 PLA2G2A (0.55) CYP1A2CYP2C19ALOX5CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102850324-A Indole compounds MICROBIA INC 2013-01-02 CN disclosed
CN-101563337-A Indole compounds MICROBIA INC (US) 2009-10-21 CN disclosed