SCHEMBL4778730

SCHEMBL4778730

CC(=O)Oc1c(C)n(Cc2nc3ccccc3s2)c2cc(F)c(C)cc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.56
CYP1A2 P05177 1/20 0.45
CYP2C19 P33261 1/20 0.45
KLKB1 P03952 1/20 0.42
KLK1 P06870 1/20 0.42
P2RX7 Q99572 1/20 0.41
AKR1B1 P15121 8/20 0.40
MAPT P10636 5/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
ALDH1A1 P00352 3/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
POLB P06746 1/20 0.38
HTT P42858 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27768505 0.91 PTGDR2 (0.53) PTGDR2CYP1A2CYP2C19KLKB1KLK1
SCHEMBL4777221 0.89 PTGDR2 (0.70) PTGDR2CYP1A2CYP2C19KLKB1KLK1
SCHEMBL27768408 0.85 PTGDR2 (0.52) PTGDR2CYP1A2CYP2C19KLKB1KLK1
SCHEMBL27789966 0.85 PTGDR2 (0.56) PTGDR2CYP1A2CYP2C19KLKB1KLK1
SCHEMBL27790170 0.84 PTGDR2 (0.50) PTGDR2CYP1A2CYP2C19KLKB1KLK1
SCHEMBL27905712 0.83 PTGDR2 (0.49) PTGDR2CYP1A2CYP2C19KLKB1KLK1
SCHEMBL27768501 0.83 PTGDR2 (0.56) PTGDR2CYP1A2CYP2C19KLKB1KLK1
SCHEMBL2000681 0.82 PTGDR2 (0.79) PTGDR2AKR1B1
SCHEMBL2007317 0.74 PTGDR2 (0.73) PTGDR2CYP1A2CYP2C19AKR1B1KDM4E
SCHEMBL2010037 0.73 PTGDR2 (0.72) PTGDR2CYP1A2CYP2C19KLKB1KLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102850324-A Indole compounds MICROBIA INC 2013-01-02 CN disclosed
CN-101563337-A Indole compounds MICROBIA INC (US) 2009-10-21 CN disclosed
EP-1931632-A2 USEFUL INDOLE COMPOUNDS Microbia Inc. (US) 2008-06-18 EP disclosed
WO-2007022501-A2 USEFUL INDOLE COMPOUNDS MICROBIA, INC. (US) 2007-02-22 WO disclosed