SCHEMBL27768446

SCHEMBL27768446

O=C(c1cn(-c2cccnc2)nn1)c1cn(-c2cccnc2)nn1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESRRA P11474 13/20 0.51
MIF P14174 1/20 0.48
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA4 P22748 2/20 0.47
CA9 Q16790 2/20 0.47
CYP2A6 P11509 1/20 0.44
GRM5 P41594 1/20 0.43
GRM1 Q13255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL71218 0.89 ESRRA (0.47) ESRRAMIFCA1CA2CA4
SCHEMBL30398916 0.88 ESRRA (0.46) ESRRAMIFCA1CA2CA4
SCHEMBL12571597 0.84 CA12 (0.55) ESRRAMIFCA1CA2CA9
SCHEMBL27768462 0.81 ESRRA (0.71) ESRRACA1CA2CA4CA9
SCHEMBL2113115 0.81 NPC1 (0.51) ESRRACA1CA2CA4CA9
SCHEMBL1083385 0.81 ESRRA (0.43) ESRRAMIFCA1CA2CA4
SCHEMBL71676 0.80 RIPK1 (0.49) MIF
SCHEMBL27768480 0.80 ESRRA (0.53) ESRRACA1CA2CA4CA9
SCHEMBL369905 0.76 MIF (0.44) MIFCA1CA2CA9CYP2A6
SCHEMBL368478 0.76 DDT (0.47) MIFGRM5GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102850324-A Indole compounds MICROBIA INC 2013-01-02 CN disclosed
CN-101563337-A Indole compounds MICROBIA INC (US) 2009-10-21 CN disclosed