SCHEMBL27769050

SCHEMBL27769050

COC(=O)c1ccc(-c2cccc(F)c2)s1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESRRG P62508 8/20 0.59
TP53 P04637 3/20 0.56
MAPT P10636 1/20 0.56
RPS6KB1 P23443 1/20 0.54
CSNK1D P48730 1/20 0.54
GSK3A P49840 1/20 0.54
GSK3B P49841 1/20 0.54
DYRK1A Q13627 1/20 0.54
NTRK2 Q16620 1/20 0.54
AURKB Q96GD4 1/20 0.54
ESR1 P03372 3/20 0.53
ESR2 Q92731 2/20 0.53
HSD17B1 P14061 2/20 0.53
HSD17B2 P37059 2/20 0.53
HDAC6 Q9UBN7 1/20 0.52
HPGDS O60760 1/20 0.50
ACKR3 P25106 1/20 0.49
KDM4E B2RXH2 1/20 0.49
NPC1 O15118 1/20 0.49
ALDH1A1 P00352 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6805238 0.84 KDM4E (0.67) ESRRGMAPTESR1ESR2HSD17B1
SCHEMBL3749139 0.84 HPGDS (0.69) ESRRGTP53MAPTESR1ESR2
SCHEMBL71536 0.84 RAB9A (0.66) TP53MAPTHSD17B1HSD17B2HDAC6
SCHEMBL13525288 0.84 HSD17B1 (0.59) ESRRGTP53MAPTESR1ESR2
SCHEMBL3918681 0.82 HPGDS (0.59) ESRRGTP53MAPTESR1ESR2
SCHEMBL6477476 0.82 KDM4E (0.58) ESRRGTP53MAPTHSD17B1HSD17B2
SCHEMBL2491378 0.81 RAB9A (0.72) ESRRGTP53MAPTHSD17B1HSD17B2
SCHEMBL27565420 0.80 ESRRG (0.59) ESRRGTP53MAPTRPS6KB1CSNK1D
SCHEMBL13524643 0.80 HPGDS (0.48) TP53GSK3AGSK3BAURKBHSD17B1
SCHEMBL17208107 0.80 HSD17B1 (0.56) ESRRGMAPTRPS6KB1CSNK1DGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100584840-C Substituted heterocyclic compounds and uses thereof ASTRAZENECA AB 2010-01-27 CN disclosed