SCHEMBL27769345

SCHEMBL27769345

CCc1nnnn1-c1cc(-c2ccccc2)c(Cl)c(C(=O)O)c1C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
HSD11B1 P28845 1/20 0.39
KCNN4 O15554 1/20 0.35
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
DHODH Q02127 1/20 0.35
FABP3 P05413 1/20 0.35
FABP4 P15090 1/20 0.35
FABP5 Q01469 1/20 0.35
TP53 P04637 1/20 0.35
TSHR P16473 2/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TACR1 P25103 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27925737 0.91 NPC1 (0.39) NPC1HSD11B1KCNN4FABP3FABP4
SCHEMBL27769320 0.89 KCNN4 (0.38) NPC1HSD11B1KCNN4DHODHFABP3
SCHEMBL27769411 0.89 KCNN4 (0.41) NPC1HSD11B1KCNN4PDCD1CD274
SCHEMBL27769319 0.86 ALDH1A1 (0.42) TP53ALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL27748148 0.86 KCNN4 (0.37) NPC1HSD11B1KCNN4PDCD1CD274
SCHEMBL27748171 0.78 TRPV1 (0.36) HSD11B1KCNN4TP53ALDH1A1LMNA
SCHEMBL16875748 0.77 NPC1 (0.43) NPC1HSD11B1DHODHTP53TSHR
SCHEMBL27769340 0.76 KCNN4 (0.37) NPC1KCNN4DHODHTSHRALDH1A1
SCHEMBL27748143 0.76 AKR1C2 (0.40) NPC1HSD11B1TP53ALDH1A1MEN1
SCHEMBL27769338 0.75 ALDH1A1 (0.39) KCNN4DHODHTSHRALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101479250-B Tetrazole-substituted arylamides HOFFMANN LA ROCHE 2013-05-22 CN disclosed
CN-101479250-A Tetrazole-substituted arylamides HOFFMANN LA ROCHE (CH) 2009-07-08 CN disclosed