SCHEMBL27769320

SCHEMBL27769320

CCc1nnnn1-c1cc(-c2ccccc2)c(Cl)c(C(=O)O)c1F

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 2/20 0.38
NPC1 O15118 1/20 0.38
HSD11B1 P28845 2/20 0.37
CDK1 P06493 1/20 0.37
CDK2 P24941 1/20 0.37
GSK3B P49841 1/20 0.37
DHODH Q02127 1/20 0.36
TP53 P04637 2/20 0.35
FABP3 P05413 1/20 0.35
FABP4 P15090 1/20 0.35
FABP5 Q01469 1/20 0.35
ALDH1A1 P00352 2/20 0.34
MAPK1 P28482 1/20 0.34
P2RX7 Q99572 1/20 0.33
FAAH O00519 1/20 0.33
MGLL Q99685 1/20 0.33
MDM2 Q00987 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27748148 0.93 KCNN4 (0.37) KCNN4NPC1HSD11B1CDK1CDK2
SCHEMBL27925737 0.91 NPC1 (0.39) KCNN4NPC1HSD11B1TP53FABP3
SCHEMBL27769345 0.89 NPC1 (0.40) KCNN4NPC1HSD11B1DHODHTP53
SCHEMBL27748171 0.89 TRPV1 (0.36) KCNN4HSD11B1CDK1CDK2GSK3B
SCHEMBL27769411 0.87 KCNN4 (0.41) KCNN4NPC1HSD11B1DHODHTP53
SCHEMBL27769340 0.85 KCNN4 (0.37) KCNN4NPC1DHODHALDH1A1MDM2
SCHEMBL27769329 0.81 ALDH1A1 (0.36) KCNN4ALDH1A1MAPK1
SCHEMBL27748146 0.80 FABP4 (0.36) KCNN4TP53FABP4FABP5ALDH1A1
SCHEMBL16875757 0.78 ALDH1A1 (0.38) KCNN4NPC1HSD11B1DHODHALDH1A1
SCHEMBL27748142 0.78 KCNN4 (0.36) KCNN4DHODHALDH1A1MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101479250-B Tetrazole-substituted arylamides HOFFMANN LA ROCHE 2013-05-22 CN disclosed
CN-101479250-A Tetrazole-substituted arylamides HOFFMANN LA ROCHE (CH) 2009-07-08 CN disclosed