SCHEMBL27770205

SCHEMBL27770205

C[C](C)Cc1ccc2c(C3CCCCC3)c(Br)[nH]c2c1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
KCNH2 Q12809 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
HDAC1 Q13547 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HPGD P15428 1/20 0.31
NQO1 P15559 1/20 0.30
KIF11 P52732 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27711877 0.86 KDM4E (0.44) MEN1KMT2AALDH1A1KDM4EHPGD
SCHEMBL84762 0.80 MAOA (0.33) HTR2AHTR2CKCNH2ALDH1A1KDM4E
SCHEMBL803700 0.78 NPC1 (0.48) HTR2AHTR2CKCNH2KMT2AALDH1A1
SCHEMBL13286195 0.78 KIF11 (0.41) MEN1KMT2AALDH1A1KDM4EKIF11
SCHEMBL27791475 0.77 S1PR1 (0.32) HTR2AHTR2CKCNH2
SCHEMBL13792682 0.75 KDM4E (0.49) ALDH1A1KDM4EHPGD
SCHEMBL50743 0.74 PARP1 (0.46) KMT2AALDH1A1KDM4EHPGDKIF11
SCHEMBL13965805 0.73 CCNA2 (0.36) MEN1KMT2AALDH1A1KDM4EHPGD
SCHEMBL18661421 0.73 CHEK2 (0.42) MEN1KMT2AALDH1A1KDM4E
SCHEMBL50237 0.72 PARP1 (0.50) MEN1KMT2AALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101918406-B Compounds for the treatment of hepatitis c BRISTOL MYERS SQUIBB CO 2013-04-17 CN disclosed
CN-101918410-B Cyclopropyl fused indolobenzazepine HCV NS5B inhibitors BRISTOL MYERS SQUIBB CO 2013-02-27 CN disclosed
CN-101679441-B Compounds for the treatment of hepatitis c BRISTOL MYERS SQUIBB CO 2012-11-14 CN disclosed
CN-101730698-B Compounds for the treatment of hepatitis c BRISTOL MYERS SQUIBB CO 2012-09-05 CN disclosed
CN-101631790-B Compounds for the treatment of hepatitis c BRISTOL MYERS SQUIBB CO 2012-07-18 CN disclosed
CN-101730698-A Compounds for the treatment of hepatitis c BRISTOL MYERS SQUIBB CO 2010-06-09 CN disclosed
CN-101679442-A The compound that is used for the treatment of hepatitis C BRISTOL MYERS SQUIBB CO 2010-03-24 CN disclosed
CN-101679441-A Compounds for the treatment of hepatitis c BRISTOL MYERS SQUIBB CO 2010-03-24 CN disclosed
CN-101657455-A Compounds for the treatment of hepatitis C SQUIBB BRISTOL MYERS CO US 2010-02-24 CN disclosed
CN-101646674-A The indoles and the benzoazepine derivative that are used for the treatment of hepatitis C SQUIBB BRISTOL MYERS CO US 2010-02-10 CN disclosed
CN-101631790-A The compound that is used for the treatment of hepatitis C BRISTOL MYERS SQUIBB CO 2010-01-20 CN disclosed