SCHEMBL27770362

SCHEMBL27770362

COCCN1C(c2ccc(Cl)cc2)=NNC1C=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APOBEC3G Q9HC16 1/20 0.37
ALDH1A1 P00352 7/20 0.35
CYP1A2 P05177 5/20 0.35
CYP3A4 P08684 4/20 0.35
CYP2C9 P11712 4/20 0.35
HSD17B10 Q99714 4/20 0.35
CASP1 P29466 4/20 0.35
CASP7 P55210 4/20 0.35
TSHR P16473 3/20 0.35
ALOX15 P16050 2/20 0.35
HPGD P15428 2/20 0.35
CYP2C19 P33261 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
CYP2D6 P10635 2/20 0.34
MAPK11 Q15759 1/20 0.34
MAPK14 Q16539 1/20 0.34
USP2 O75604 3/20 0.33
HIF1A Q16665 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27848965 0.80 HDAC1 (0.32) L3MBTL1
SCHEMBL27909622 0.80 TP53 (0.41) ALDH1A1CYP1A2CYP3A4CYP2C9TSHR
SCHEMBL27770365 0.78 ALDH1A1 (0.35) ALDH1A1HSD17B10HPGDL3MBTL1USP2
SCHEMBL27909686 0.73
SCHEMBL27770355 0.73
SCHEMBL28027065 0.72 GAA (0.36)
SCHEMBL27770358 0.69 PDE4A (0.32) MEN1KMT2A
SCHEMBL27515004 0.64 SMN1; SMN2 (0.41) ALDH1A1HPGDKMT2ALMNAKDM4E
SCHEMBL28058563 0.64 MAOA (0.32) ALDH1A1L3MBTL1KMT2ALMNA
SCHEMBL27561988 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101495458-B Substituted arylimidazolone and triazolone as inhibitors of vasopressin receptors BAYER IP GMBH 2014-01-29 CN disclosed
CN-101495458-A Substituted arylimidazolone and triazolone as inhibitors of vasopressin receptors BAYER HEALTHCARE AG (DE) 2009-07-29 CN disclosed