SCHEMBL27770502

SCHEMBL27770502

NCc1c(Cl)cccc1NS(=O)(=O)c1ccc(F)cc1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.67
MEN1 O00255 1/20 0.67
KMT2A Q03164 1/20 0.67
KEAP1 Q14145 1/20 0.50
NFE2L2 Q16236 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
CCR2 P41597 1/20 0.48
GLO1 Q04760 1/20 0.48
STAT3 P40763 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27749430 0.86 LMNA (0.54) TSHRMEN1KMT2AKEAP1NFE2L2
SCHEMBL27858487 0.83 KDM4E (0.54) TSHRMEN1KMT2ACCR2
SCHEMBL2175966 0.78 TSHR (0.72) TSHRMEN1KMT2AKEAP1NFE2L2
SCHEMBL3980968 0.75 MEN1 (0.67) TSHRMEN1KMT2A
SCHEMBL7589375 0.75 MEN1 (0.77) TSHRMEN1KMT2AKEAP1NFE2L2
SCHEMBL29833597 0.73 ALDH1A1 (0.55) TSHRMEN1KMT2AKEAP1NFE2L2
SCHEMBL12407080 0.73 LMNA (0.55) TSHRMEN1KMT2AKEAP1NFE2L2
SCHEMBL28728692 0.73 ALDH1A1 (0.55) TSHRMEN1KMT2AKEAP1NFE2L2
SCHEMBL21497038 0.72 KMT2A (0.59) TSHRMEN1KMT2A
SCHEMBL1471525 0.72 MEN1 (0.62) TSHRMEN1KMT2ASTAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101500554-B Sulfonamide compound or salt thereof ASTELLAS PHARMA INC 2012-06-27 CN disclosed
CN-101500554-A Sulfonamide compound or salt thereof ASTELLAS PHARMA INC (JP) 2009-08-05 CN disclosed