SCHEMBL27770608

SCHEMBL27770608

CCP(=O)(CC)OC(F)(F)C(F)(F)c1cccc(N)c1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.45
MAPK1 P28482 1/20 0.45
CYP3A4 P08684 2/20 0.35
TP53 P04637 1/20 0.35
PTGS1 P23219 3/20 0.35
KDM4E B2RXH2 2/20 0.33
PGK1 P00558 1/20 0.33
PGK2 P07205 1/20 0.33
PTPN1 P18031 1/20 0.32
CCNT1 O60563 2/20 0.32
CDK9 P50750 2/20 0.32
ALDH1A1 P00352 2/20 0.31
MAOB P27338 1/20 0.31
ACP3 P15309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27749823 0.80 TRPA1 (0.40) CYP3A4ALDH1A1
SCHEMBL27770581 0.79 PTPRC (0.48) TSHRCCNT1CDK9ALDH1A1
SCHEMBL642678 0.74 TSHR (0.45) TSHRMAPK1CYP3A4TP53PTGS1
SCHEMBL10128394 0.73 TSHR (0.44) TSHRMAPK1CYP3A4TP53PTGS1
SCHEMBL10714404 0.72 TSHR (0.74) TSHRMAPK1CYP3A4PTGS1KDM4E
SCHEMBL642679 0.71 TSHR (0.39) TSHRMAPK1TP53PTGS1KDM4E
SCHEMBL642867 0.71 TSHR (0.47) TSHRMAPK1CYP3A4TP53PTGS1
SCHEMBL7586287 0.69 TSHR (0.63) TSHRMAPK1CYP3A4PTGS1PGK1
SCHEMBL27770580 0.69 ALDH1A1 (0.43) TSHRMAPK1CYP3A4KDM4EALDH1A1
SCHEMBL3843446 0.69 TSHR (0.68) TSHRMAPK1CYP3A4PTGS1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101501051-A Amides as sphingomyeline inhibitors NOVARTIS AG (CH) 2009-08-05 CN disclosed