SCHEMBL27770667

SCHEMBL27770667

Clc1ccccc1-c1cnc(CCBr)s1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LIMK1 P53667 13/20 0.43
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
AVPR2 P30518 1/20 0.39
AVPR1A P37288 1/20 0.39
MAPK14 Q16539 3/20 0.36
LIMK2 P53671 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2441087 0.87 LIMK1 (0.44) LIMK1HDAC1HDAC6AVPR2AVPR1A
SCHEMBL28815683 0.77 LOXL2 (0.55)
SCHEMBL2443835 0.73 CTSA (0.36) LIMK1AVPR2AVPR1A
SCHEMBL2440919 0.71 LIMK1 (0.48) LIMK1HDAC1HDAC6MAPK14
SCHEMBL38544 0.71 LIMK1 (0.72) LIMK1HDAC1HDAC6MAPK14KDM4E
SCHEMBL30513213 0.71 LIMK1 (0.72) LIMK1HDAC1HDAC6MAPK14KDM4E
SCHEMBL16513196 0.71 LIMK1 (0.43) LIMK1HDAC1HDAC6MAPK14LIMK2
SCHEMBL16513199 0.71 LIMK1 (0.64) LIMK1LIMK2
SCHEMBL28781561 0.70 LIMK1 (0.43) LIMK1HDAC1HDAC6MAPK14LIMK2
SCHEMBL16513235 0.69 LIMK1 (0.41) LIMK1HDAC1HDAC6AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101646660-A Compounds and methods for modulating G protein-coupled receptors IRM LLC VG 2010-02-10 CN disclosed