SCHEMBL2777086

SCHEMBL2777086

CC(C)[C@H](NC(=O)O)C(=O)N1CCC(Oc2cccnc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.53
ALDH1A1 P00352 3/20 0.52
CCR1 P32246 5/20 0.46
HTT P42858 1/20 0.45
SPR P35270 1/20 0.45
PREP P48147 1/20 0.43
MAPT P10636 1/20 0.43
NAMPT P43490 2/20 0.43
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2774368 0.87 EPHX2 (0.50) EPHX2ALDH1A1CCR1PREPMAPT
SCHEMBL2776309 0.86 ACACB (0.46) ALDH1A1CCR1MAPTNAMPT
SCHEMBL2777506 0.85 ALDH1A1 (0.44) EPHX2ALDH1A1CCR1PREPKCNH2
SCHEMBL2774934 0.83 CCR1 (0.46) ALDH1A1CCR1KCNH2
SCHEMBL2775312 0.82 ALDH1A1 (0.47) EPHX2ALDH1A1CCR1HTTSPR
SCHEMBL2775675 0.82 EPHX2 (0.52) EPHX2ALDH1A1HTTSPRMAPT
SCHEMBL2779095 0.82 CCR1 (0.48) CCR1KCNH2
SCHEMBL2776130 0.82 GPR119 (0.50) ALDH1A1CCR1
SCHEMBL2774679 0.82 EPHX2 (0.51) EPHX2ALDH1A1CCR1NAMPTKCNH2
Hydrochloric Acid SCHEMBL2775304 0.81 EPHX2 (0.51) EPHX2ALDH1A1HTTSPRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2258697-A1 HYDROXYQUINOXALINECARBOXAMIDE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2010-12-08 EP disclosed