SCHEMBL2774679

SCHEMBL2774679

CC(C)[C@H](NC(=O)O)C(=O)N1CCC(Oc2cnccn2)CC1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.51
CYP2C9 P11712 1/20 0.50
NAAA Q02083 9/20 0.46
ACACB O00763 1/20 0.41
NAMPT P43490 2/20 0.41
ALDH1A1 P00352 1/20 0.40
CCR1 P32246 4/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2775696 0.85 EPHX2 (0.53) EPHX2NAMPTALDH1A1CCR1KCNH2
SCHEMBL2780460 0.83 NAMPT (0.49) ACACBNAMPTCCR1KCNH2
SCHEMBL2776473 0.82 GPR119 (0.44) CCR1KCNH2
SCHEMBL2777086 0.82 EPHX2 (0.53) EPHX2NAMPTALDH1A1CCR1KCNH2
Hydrochloric Acid SCHEMBL2773858 0.81 EPHX2 (0.48) EPHX2CYP2C9NAAAACACBNAMPT
SCHEMBL2774368 0.81 EPHX2 (0.50) EPHX2CYP2C9ACACBNAMPTALDH1A1
SCHEMBL2776856 0.81 MMP1 (0.59) NAMPTCCR1KCNH2
SCHEMBL2776032 0.81 NAMPT (0.50) EPHX2CYP2C9NAMPTCCR1
SCHEMBL2774593 0.81 EPHX2 (0.46) EPHX2CYP2C9NAAANAMPTALDH1A1
SCHEMBL2777388 0.80 KMT2A (0.43) NAMPTCCR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2258697-A1 HYDROXYQUINOXALINECARBOXAMIDE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2010-12-08 EP disclosed