SCHEMBL27775498

SCHEMBL27775498

Cc1cc(-c2ccc(O)cc2)ncc1[N+](=O)[O-]

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
MAPT P10636 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
LDHA P00338 1/20 0.41
TSHR P16473 2/20 0.40
GPR35 Q9HC97 2/20 0.39
ELANE P08246 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ALOX5 P09917 1/20 0.37
DYRK1A Q13627 1/20 0.37
DYRK1B Q9Y463 1/20 0.37
ALKBH5 Q6P6C2 1/20 0.37
FTO Q9C0B1 1/20 0.37
ERN1 O75460 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2810982 0.84 LDHA (0.54) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL14689223 0.78 CYP2A6 (0.53) MAPTCYP2C9CYP2C19MEN1KMT2A
SCHEMBL27775500 0.77 KMT2A (0.51) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL16701399 0.76 TSHR (0.53) ALDH1A1MAPTTSHRGPR35MEN1
SCHEMBL801081 0.75 ALDH1A1 (0.49) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL1762742 0.75 TSHR (0.47) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL29697302 0.74 ERN1 (0.48) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL29838652 0.72 AAK1 (0.48) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL31436939 0.72 ALDH1A1 (0.53) ALDH1A1MAPTTSHRGPR35MEN1
SCHEMBL27775497 0.72 ALDH1A1 (0.43) ALDH1A1MAPTTSHRGPR35ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101511813-B Heterocyclic FXR binding compounds PHENEX PHARMACEUTICALS AG 2012-12-12 CN disclosed
CN-101511813-A Heterocyclic FXR binding compounds PHENEX PHARMACEUTICALS AG (DE) 2009-08-19 CN disclosed