SCHEMBL27775801

SCHEMBL27775801

CP(C)(=O)OCC(=O)c1cc(F)ccc1C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.37
KCNK9 Q9NPC2 1/20 0.37
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
CES2 O00748 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
EPHX2 P34913 1/20 0.35
PPARG P37231 1/20 0.35
P2RX1 P51575 1/20 0.35
TMPRSS4 Q9NRS4 1/20 0.35
MAPT P10636 2/20 0.34
KMT2A Q03164 2/20 0.34
HTT P42858 2/20 0.34
IDO1 P14902 1/20 0.34
MEN1 O00255 1/20 0.34
PKM P14618 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
CHRM5 P08912 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27775828 0.89 KMT2A (0.40) KCNK3KCNK9HCRTR1HCRTR2CES2
SCHEMBL27755386 0.85 HTT (0.46) LMNATMPRSS4MAPTHTTRAB9A
SCHEMBL27755234 0.78 NPC1 (0.39) CES2MAPTKMT2AHTTMEN1
SCHEMBL2325106 0.78 EPHX2 (0.38) KCNK3KCNK9HCRTR1HCRTR2CES2
SCHEMBL2325110 0.77 KCNK3 (0.37) KCNK3KCNK9HCRTR1HCRTR2CES2
SCHEMBL26020578 0.77 CES2 (0.43) KCNK3KCNK9HCRTR1HCRTR2CES2
SCHEMBL27775993 0.77 HPGD (0.44) MAPTKMT2ANPC1RAB9A
SCHEMBL16914396 0.74 PTPN1 (0.47) HCRTR1HCRTR2CES2LMNAGAA
SCHEMBL27776094 0.72 NPC1 (0.48) CES2LMNAMAPTPKMNPC1
SCHEMBL27755344 0.72 SLC6A2 (0.38) CES2LMNAGAAP2RX1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101528713-A Pyridazine derivatives as inhibitors of 11 beta-hydroxysteroid dehydrogenase type 1 HOFFMANN LA ROCHE (CH) 2009-09-09 CN disclosed