SCHEMBL27780658

SCHEMBL27780658

CCCCc1nc2cccc(C)c2c(=O)n1N1CCCCC1C(=O)C=O

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
LMNA P02545 3/20 0.38
KCNK3 O14649 1/20 0.38
HTR1A P08908 1/20 0.36
PIK3CD O00329 2/20 0.36
HRH3 Q9Y5N1 1/20 0.35
ELANE P08246 5/20 0.34
CNR2 P34972 2/20 0.34
RECQL P46063 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27759268 0.85 HRH3 (0.40) KCNH2CYP3A4CYP2D6LMNAKCNK3
SCHEMBL27780650 0.81 GAA (0.37) LMNAKCNK3PIK3CDHRH3ELANE
SCHEMBL27759292 0.76 HRH3 (0.42) KCNH2CYP3A4LMNAPIK3CDHRH3
SCHEMBL27759300 0.76 HRH3 (0.42) KCNH2PIK3CDHRH3
SCHEMBL27780676 0.76 TNF (0.42) KCNH2LMNAKCNK3PIK3CDHRH3
SCHEMBL27780703 0.75 USP2 (0.37) KCNH2CYP3A4CYP2D6LMNAKCNK3
SCHEMBL27759279 0.74 LMNA (0.31) LMNA
SCHEMBL28030923 0.73 HDAC1 (0.38) LMNAHTR1APIK3CDELANECNR2
SCHEMBL24113864 0.66 PIK3CD (0.39) LMNAHTR1APIK3CDELANESMN1; SMN2
SCHEMBL7421353 0.65 PPARG (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101535291-A 5-substituted quinazolinone derivatives as antitumor agents CELGENE CORP (US) 2009-09-16 CN disclosed