SCHEMBL28030923

SCHEMBL28030923

CCCCc1nc2cccc(C)c2c(=O)n1C1CCC(C(=O)C=O)NC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 6/20 0.38
PIK3CD O00329 1/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPK1 P28482 2/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HTR1A P08908 1/20 0.34
LMNA P02545 2/20 0.33
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
ELANE P08246 2/20 0.32
MEN1 O00255 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
AGTR1 P30556 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28030321 0.92 PIK3CD (0.36) PIK3CD
SCHEMBL28030946 0.85 DDB1 (0.39) PIK3CDALDH1A1MAPK1NPSR1LMNA
SCHEMBL16597161 0.76 ALDH1A1 (0.48) PIK3CDALDH1A1MAPK1MAPTSMN1; SMN2
SCHEMBL27936623 0.76 DDB1 (0.51) PIK3CDALDH1A1MAPK1NPSR1LMNA
SCHEMBL28822138 0.76 HRH3 (0.39) PIK3CD
SCHEMBL25346369 0.76 TNF (0.34) ALDH1A1MAPK1NPSR1KMT2A
SCHEMBL28030943 0.76 DDB1 (0.38) ALDH1A1MAPK1NPSR1KMT2A
SCHEMBL28030926 0.76 USP2 (0.38) ELANE
SCHEMBL27759269 0.73 CNR2 (0.38) ALDH1A1NPSR1CNR2MEN1HTT
SCHEMBL16584875 0.73 SMN1; SMN2 (0.41) PIK3CDMAPTSMN1; SMN2NPSR1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105017212-A 5-substituted quinazolinone derivatives using as antineoplastic agent CELGENE CORP 2015-11-04 CN disclosed
CN-104910133-A 5-SUBSTITUTED QUINAZOLINONE DERIVATIVES AS ANTITUMOR AGENTS CELGENE CORP 2015-09-16 CN disclosed
CN-104876908-A 5-substituted quinazolinone derivatives as anti-cancer agents CELGENE CORP 2015-09-02 CN disclosed