SCHEMBL27787604

SCHEMBL27787604

[CH2]CCNC(=O)C(Br)CC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 2/20 0.45
TSHR P16473 1/20 0.45
KMT2A Q03164 3/20 0.38
ALDH1A1 P00352 3/20 0.38
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC11 Q96DB2 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
HDAC9 Q9UKV0 1/20 0.32
HDAC5 Q9UQL6 1/20 0.32
DPP7 Q9UHL4 2/20 0.32
MEN1 O00255 2/20 0.31
MAPT P10636 1/20 0.31
ALDH1A2 O94788 1/20 0.30
ALDH2 P05091 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1772263 0.78
SCHEMBL9036061 0.77 TSHR (0.46) USP2TSHRKMT2AMEN1
SCHEMBL28580193 0.76 EPHX1 (0.55) DPP7
SCHEMBL8212374 0.76 GNAI3 (0.46) USP2TSHRKMT2AALDH1A1DPP7
SCHEMBL28559240 0.76 EPHX1 (0.55) DPP7
SCHEMBL27340657 0.75 TSHR (0.41) USP2TSHRKMT2AALDH1A1MEN1
SCHEMBL11202268 0.73 ALDH1A1 (0.42) USP2TSHRKMT2AALDH1A1MAPT
SCHEMBL843281 0.73
SCHEMBL8083315 0.72 CYP2C19 (0.48) USP2TSHRKMT2AALDH1A1MEN1
SCHEMBL6272869 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101600698-B Quinazolinone and isoquinolinone acetamide derivatives ORGANON NV 2012-01-11 CN disclosed
CN-101600698-A Quinazolinone and isoquinolinone acetamide derivatives ORGANON NV (NL) 2009-12-09 CN disclosed