SCHEMBL27796334

SCHEMBL27796334

N#Cc1c(N)n(OC(=O)c2ccccc2)c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
STAT3 P40763 2/20 0.43
MAPK1 P28482 1/20 0.43
ELANE P08246 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
CCR2 P41597 1/20 0.38
TSHR P16473 2/20 0.37
KMT2A Q03164 6/20 0.37
MEN1 O00255 4/20 0.37
GAA P10253 3/20 0.37
KDM4E B2RXH2 3/20 0.37
GLA P06280 2/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
PKM P14618 1/20 0.36
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
EGFR P00533 1/20 0.35
SRC P12931 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27800832 0.77 F2 (0.48) ALDH1A1MAPK1ELANETDP1TSHR
SCHEMBL27796324 0.69 STAT3 (0.52) ALDH1A1STAT3ELANETDP1TSHR
SCHEMBL28702396 0.68 KMT2A (0.40) ALDH1A1ELANETDP1KMT2AKDM4E
SCHEMBL5199685 0.68 ALDH1A1 (0.46) ALDH1A1STAT3MAPK1TDP1TSHR
SCHEMBL7488560 0.67 KDM4E (0.57) ALDH1A1STAT3MAPK1TDP1TSHR
SCHEMBL29057689 0.67 KDM4E (0.49) ALDH1A1TDP1KMT2AMEN1GAA
SCHEMBL9381587 0.66 EGFR (0.62) ALDH1A1MAPK1TDP1TSHRKMT2A
SCHEMBL9022394 0.66 ALDH1A1 (0.47) ALDH1A1STAT3MAPK1ELANETDP1
SCHEMBL2238063 0.65 LMNA (0.54) ALDH1A1MAPK1TDP1TSHRKMT2A
SCHEMBL28691611 0.64 CYP11B1 (0.41) ALDH1A1KMT2AMEN1EGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101679251-B (Aza)indole derivative and use thereof for medical purposes KISSEI PHARMACEUTICAL 2013-10-02 CN disclosed
CN-101679251-A (Aza)indole derivative and use thereof for medical purposes KISSEI PHARMACEUTICAL 2010-03-24 CN disclosed