SCHEMBL27799415

SCHEMBL27799415

NC(=O)c1ccc2c(c1)CCN=C2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.40
SIRT2 Q8IXJ6 2/20 0.38
TSHR P16473 1/20 0.38
HSD17B3 P37058 1/20 0.37
NNMT P40261 3/20 0.36
LCK P06239 1/20 0.36
HDAC1 Q13547 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HDAC3 O15379 1/20 0.35
CYP2C19 P33261 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27576919 0.87 KDM1A (0.41) KDM1ASIRT2TSHRHSD17B3NNMT
Hydrochloric Acid SCHEMBL27985832 0.85 KDM1A (0.40) KDM1ASIRT2TSHRHSD17B3NNMT
SCHEMBL27918521 0.85 ALDH1A1 (0.49) KDM1ATSHRCYP2C19KDM4EALDH1A1
SCHEMBL27774598 0.83 PRSS1 (0.38)
SCHEMBL16038861 0.75 NPC1 (0.47) KDM1AHDAC1HDAC8HDAC6HDAC2
SCHEMBL29769963 0.73 CASP1 (0.37) KDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL9573469 0.73 DRD2 (0.37) HSD17B10
SCHEMBL7341198 0.72 KDM1A (0.40) KDM1ATSHRHSD17B3NNMTLCK
SCHEMBL27914874 0.71 ALDH1A1 (0.49) KDM1ATSHRCYP2C19KDM4EALDH1A1
SCHEMBL27556733 0.71 KDM1A (0.39) KDM1ATSHRHSD17B3NNMTLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814040-A Fused 1,4-dihydrodioxin derivatives as inhibitors of heat shock transcription factor 1 癌症研究科技有限公司 2016-07-27 CN disclosed
CN-101679273-A 1-substituted tetrahydroisoquinoline compound ASTELLAS PHARMA INC 2010-03-24 CN disclosed