SCHEMBL27801367

SCHEMBL27801367

NC=CCS(=O)(=O)NC(CNC(=O)c1ccc2cccc(-c3cccc4ccccc34)c2n1)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.36
ITGAV P06756 9/20 0.36
ITGB3 P05106 4/20 0.36
ITGA2B P08514 3/20 0.36
FDPS P14324 1/20 0.34
GAA P10253 1/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
PGGT1B P53609 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2117513 0.87 ITGAV (0.39) CASP1ITGAVITGB3ITGA2BFDPS
SCHEMBL27801369 0.83 CASP1 (0.36) CASP1ITGAVITGB3ITGA2BFDPS
SCHEMBL2116269 0.77 FDPS (0.39) FDPSGAAFNTAPGGT1B
Hydrochloric Acid SCHEMBL2116377 0.76 FDPS (0.38) FDPSGAAFNTAPGGT1B
SCHEMBL2119125 0.72 FDPS (0.42) FDPSGAAFNTAPGGT1B
Ammonia Solution, Strong SCHEMBL2117519 0.72 GAA (0.36) FDPSGAA
Hydrochloric Acid SCHEMBL2119121 0.71 FDPS (0.42) FDPSGAAFNTAPGGT1B
SCHEMBL2116667 0.70 CA12 (0.38) CASP1FDPSFNTAPGGT1B
SCHEMBL2116709 0.70 HDAC8 (0.39) FDPSGAA
SCHEMBL2115818 0.70 KYNU (0.45) CASP1FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101959865-A Quinolines as farnesyl pyrophosphate synthase inhibitor NOVARTIS AG 2011-01-26 CN claimed
CN-101959865-A Quinolines as farnesyl pyrophosphate synthase inhibitor NOVARTIS AG 2011-01-26 CN disclosed