Acetic Acid

Acetic Acid

SCHEMBL2780795

CC(=O)O.COc1cccc(OC)c1CNC(=N)Nc1ccc(C#N)cn1

nearest known ligand 0.44

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Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Acetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 8/20 0.44
HCRTR1 O43613 7/20 0.44
CYP2C8 P10632 1/20 0.44
CYP2C19 P33261 1/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ROCK2 O75116 1/20 0.41
FGFR4 P22455 1/20 0.39
IDO1 P14902 1/20 0.39
MAPK1 P28482 3/20 0.38
HIF1A Q16665 1/20 0.38
IDH1 O75874 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2780626 0.95 HCRTR1 (0.41) HCRTR2HCRTR1CYP2C8CYP2C19MEN1
Acetic Acid SCHEMBL2783102 0.94 HCRTR2 (0.42) HCRTR2HCRTR1CYP2C8CYP2C19MEN1
Acetic Acid SCHEMBL2785032 0.93 HCRTR1 (0.41) HCRTR2HCRTR1CYP2C8CYP2C19MEN1
Acetic Acid SCHEMBL2782951 0.93 MAPK1 (0.47) HCRTR2HCRTR1CYP2C8CYP2C19MEN1
SCHEMBL2780807 0.89 HCRTR1 (0.39) HCRTR2HCRTR1CYP2C8CYP2C19MEN1
SCHEMBL2782892 0.88 MAPK1 (0.46) HCRTR2HCRTR1CYP2C8CYP2C19MEN1
SCHEMBL2780680 0.88 HCRTR1 (0.39) HCRTR2HCRTR1CYP2C8CYP2C19MEN1
Acetic Acid SCHEMBL2782375 0.86 HCRTR1 (0.44) HCRTR2HCRTR1CYP2C19MEN1KMT2A
Acetic Acid SCHEMBL2781387 0.83 ROCK2 (0.49) MEN1KMT2AROCK2HIF1A
SCHEMBL2781548 0.83 NTRK1 (0.50) HCRTR2HCRTR1CYP2C8CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9296697-B2 Hetaryl-substituted guanidine compounds and use thereof as binding partners for 5-HT5-receptors ABBOTT LABORATORIES (US) 2016-03-29 US disclosed
US-20100184787-A1 Heataryl-substituted guanidine compounds and use thereof as binding partners for 5-ht5-receptors ABBVIE DEUTSCHLAND GMBH & CO KG (DE) 2010-07-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100184787-A1 Heataryl-substituted guanidine compounds and use thereof as binding partners for 5-ht5-receptors HTR5A, HTR2C, HTR1E HCRTR2 533/4885HCRTR1 651/4885CYP2C8 550/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.