SCHEMBL27820175

SCHEMBL27820175

CC(=O)Oc1nnsc1CCl

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.34
TSHR P16473 2/20 0.31
MAPT P10636 2/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPK1 P28482 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27799031 0.84 ALOX5 (0.33) ALOX5TSHR
SCHEMBL27820127 0.84 ALOX5 (0.33) ALOX5TSHR
SCHEMBL28785808 0.81 ALOX5 (0.32) ALOX5TSHRMAPTKDM4EALDH1A1
SCHEMBL27797610 0.73 TSHR (0.30) TSHR
SCHEMBL6955106 0.65
SCHEMBL27820176 0.64 GABRR1 (0.31)
SCHEMBL27797611 0.64 PTGDR2 (0.30) KDM4E
SCHEMBL27797899 0.62 TSHR (0.30) TSHR
SCHEMBL11312405 0.62
SCHEMBL27965548 0.62 HPGD (0.35) ALOX5MAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101891709-A 5-halogenated methyl-1,2,3-thiadiazole compound and preparation method and use thereof UNIV NANKAI 2010-11-24 CN claimed
CN-101891709-B 5-halogenated methyl-1,2,3-thiadiazole compound and preparation method and use thereof UNIV NANKAI 2012-11-21 CN disclosed
CN-101891709-A 5-halogenated methyl-1,2,3-thiadiazole compound and preparation method and use thereof UNIV NANKAI 2010-11-24 CN disclosed