SCHEMBL278237

SCHEMBL278237

C=CCNC(C)OC(=O)C(=C)C

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.40
ALDH1A1 P00352 2/20 0.39
THRB P10828 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL368698 0.82 ALDH1A1 (0.39) TSHRALDH1A1THRBNPSR1
SCHEMBL246672 0.79 TSHR (0.44) TSHRALDH1A1THRB
SCHEMBL5576920 0.79 TSHR (0.44) TSHRALDH1A1THRB
Hydrochloric Acid SCHEMBL23116685 0.78 TSHR (0.42) TSHRALDH1A1THRB
SCHEMBL6264346 0.78 TSHR (0.42) TSHRALDH1A1THRB
SCHEMBL278175 0.78 TSHR (0.42) TSHRALDH1A1
SCHEMBL3280963 0.78 TSHR (0.47) TSHRALDH1A1THRB
Ammonia Solution, Strong SCHEMBL7765025 0.78 TSHR (0.42) TSHRALDH1A1THRB
SCHEMBL28964247 0.78 TSHR (0.42) TSHRALDH1A1THRB
SCHEMBL556918 0.76 TSHR (0.41) TSHRALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 298 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2337554-B1 AGENT FOR FIBRES CONTAINING KERATIN, COMPRISING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER AND AT LEAST ONE SPECIFIC, ADDITIONAL FILM-FORMING ANIONIC AND/OR STABILIZING ANIONIC POLYMER HENKEL AG & CO KGAA (DE) 2016-09-07 EP claimed
US-9206552-B2 Absorbent plastic pigment with improved print density containing and recording sheet containing same INTERNATIONAL PAPER COMPANY (US) 2015-12-08 US claimed
US-8777390-B2 Ink-jet printing system with reduced nozzle clogging HEWLETT-PACKARD DEVELOPMENT COMPANY, L.P. (US) 2014-07-15 US claimed
US-20140166036-A1 TRANSFORMATION MEDIUM FOR MODELS CONTAINING KERATIN FIBERS HENKEL AG & CO. KGAA (DE) 2014-06-19 US claimed
WO-2013122756-A1 ABSORBENT PLASTIC PIGMENT WITH IMPROVED PRINT DENSITY AND RECORDING SHEET CONTAINING SAME INTERNATIONAL PAPER COMPANY (US) 2013-08-22 WO claimed
US-20130215184-A1 ABSORBENT PLASTIC PIGMENT WITH IMPROVED PRINT DENSITY AND RECORDING SHEET CONTAINING SAME INTERNATIONAL PAPER COMPANY (US) 2013-08-22 US claimed
US-20120207694-A1 AGENT FOR TREATING KERATIN-CONTAINING FIBERS, CONTAINING A NON-IONIC STARCH MODIFIED BY PROPYLENE OXIDE AND AN ANIONIC POLYMER HENKEL AG & CO. KGAA 2012-08-16 US claimed
US-8132907-B2 Image forming method FUJIFILM CORPORATION (JP) 2012-03-13 US claimed
US-20110142781-A1 AGENT FOR FIBERS CONTAINING KERATIN, COMPRISING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER AND AT LEAST ONE SPECIFIC, ADDITIONAL FILM-FORMING ANIONIC AND/OR STABILIZING ANIONIC POLYMER HENKEL AG & CO. KGAA (DE) 2011-06-16 US claimed
EP-1586454-B1 Ink-jet printing methods and systems providing improved image durability HEWLETT PACKARD DEVELOPMENT CO (US) 2010-03-03 EP claimed
US-20050206705-A1 Ink-jet imaging on offset media HEWLETT-PACKARD DEVELOPMENT COMPANY, L.P. 2005-09-22 US claimed
US-6779884-B1 Ink-jet printing methods and systems providing dry rub resistance HEWLETT-PACKARD DEVELOPMENT COMPANY, L.P. 2004-08-24 US claimed
US-20040063808-A1 Ink-jet printing methods and systems providing improved image durability HEWLETT-PACKARD DEVELOPMENT COMPANY, L.P. 2004-04-01 US claimed
EP-1403346-A1 Ink-jet printing methods and systems providing improved image durability Hewlett-Packard Development Company, L.P. (US) 2004-03-31 EP claimed
US-6423461-B1 INORGANIC POLYMER AND ORGANOMETALLIC POLYMER BLEND OF POLYFERROCENES AND POLYPHOSPHAZENES XEROX CORPORATION 2002-07-23 US claimed
US-6037091-A Carrier with ferrocene containing polymer XEROX CORPORATION (US) 2000-03-14 US claimed
US-6004712-A CORE AND THEREOVER A POLYMER OF (1) METHYLMETHACRYLATE AND A MONOALKYL AMINOALKYL METHACRYLATE, OR (2) A POLYMER OF METHYLMETHACRYLATE AND DIALKYLAMINOALKYL METHACRYLATE, TONER AND DEVELOPER XEROX CORPORATION (US) 1999-12-21 US claimed
US-5574548-A Method and device for developing with a liquid MINOLTA CAMERA KABUSHIKI KAISHA (JP) 1996-11-12 US claimed
US-4212782-A Polymers of acid addition salts of methacrylic acid and a 2-mono(lower)alkylaminoethyl methacrylate NORMAC, INC. (US) 1980-07-15 US claimed
US-3950398-A Methacrylic acid addition salt of 2-mono(lower)alkyl amino ethyl methacrylate NORMAC, INC. (US) 1976-04-13 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110142781-A1 AGENT FOR FIBERS CONTAINING KERATIN, COMPRISING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER AND AT LEAST ONE SPECIFIC, ADDITIONAL FILM-FORMING ANIONIC AND/OR STABILIZING ANIONIC POLYMER KRT18, H1-10, C9 TSHR 1658/4885ALDH1A1 2479/4885THRB 2878/4885
US-20120207694-A1 AGENT FOR TREATING KERATIN-CONTAINING FIBERS, CONTAINING A NON-IONIC STARCH MODIFIED BY PROPYLENE OXIDE AND AN ANIONIC POLYMER KRT18, F12, H1-10 TSHR 1436/4885ALDH1A1 3385/4885THRB 2114/4885
US-20140166036-A1 TRANSFORMATION MEDIUM FOR MODELS CONTAINING KERATIN FIBERS KRT18, NEFM, CUTA TSHR 1366/4885ALDH1A1 3144/4885THRB 3694/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.