SCHEMBL27827331

SCHEMBL27827331

Cc1c(N2CCN(C)CC2)c(=O)oc2cc(N(C)C)ccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 15/20 1.00
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HTT P42858 2/20 0.42
MEN1 O00255 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
KMT2A Q03164 1/20 0.42
ATM Q13315 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27806711 0.82 CCR4 (1.00) CCR4
SCHEMBL179796 0.78 CCR4 (0.64) CCR4KDM4EALDH1A1HTTMEN1
SCHEMBL29527262 0.78 CCR4 (0.64) CCR4KDM4EALDH1A1HTTMEN1
SCHEMBL10881037 0.78 CCR4 (0.62) CCR4KDM4EALDH1A1HTTGLA
SCHEMBL14160791 0.76 CCR4 (0.61) CCR4KDM4EALDH1A1HTTMEN1
SCHEMBL21457065 0.73 CCR4 (0.56) CCR4KDM4EALDH1A1HTTMEN1
SCHEMBL21457084 0.69 CCR4 (0.53) CCR4KDM4EALDH1A1HTTMEN1
SCHEMBL194522 0.69 MAOA (0.61) CCR4MAOAKDM4EALDH1A1MEN1
SCHEMBL4955063 0.69 CCR4 (0.52) CCR4KDM4EALDH1A1HTTMEN1
SCHEMBL10001285 0.68 ALDH1A1 (0.54) CCR4KDM4EALDH1A1HTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102050809-B Chemokine-like factor 1 (CKLF1)/C chemokine receptor 4 (CCR4) interaction-antagonistic 3-peperazinyl coumarin derivatives INST MATERIA MEDICA CAMS 2014-12-17 CN disclosed
CN-103446154-A Applications of coumarin derivatives in preventing and curing serious brain diseases INST MATERIA MEDICA CAMS 2013-12-18 CN disclosed
CN-102050809-A Chemokine-like factor 1 (CKLF1)/C chemokine receptor 4 (CCR4) interaction-antagonistic 3-peperazinyl coumarin derivatives INST MATERIA MEDICA CAMS 2011-05-11 CN disclosed