SCHEMBL27837686

SCHEMBL27837686

O=C1CCc2cccc(OC(F)(F)F)c2O1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.35
KIF11 P52732 1/20 0.34
DDB1 Q16531 2/20 0.34
CRBN Q96SW2 2/20 0.34
GRIA1 P42261 5/20 0.34
CACNG8 Q8WXS5 5/20 0.34
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
HTR2A P28223 1/20 0.33
CACNG2 Q9Y698 1/20 0.32
AKR1B1 P15121 1/20 0.32
OPRM1 P35372 1/20 0.32
ALDH1A1 P00352 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27855565 0.76 AADAT (0.36) KDM4EHTR2CHTR2BHTR2AAKR1B1
SCHEMBL14070903 0.73 HTR1A (0.36)
SCHEMBL31040600 0.73 MAOB (0.40) HTR2CHTR2AAKR1B1L3MBTL1
SCHEMBL11123491 0.73 HPGD (0.39) AKR1B1
SCHEMBL11122122 0.73 HPGD (0.42) AKR1B1ALDH1A1
SCHEMBL12216130 0.70 ELANE (0.35) KDM4E
SCHEMBL834241 0.69 ALDH2 (0.37) KDM4EAKR1B1ALDH1A1L3MBTL1
SCHEMBL32673059 0.69 TSHR (0.37) KDM4EAKR1B1
SCHEMBL28587199 0.69 HPGD (0.41) KDM4ECRBNAKR1B1ALDH1A1
SCHEMBL16283615 0.69 PTGS1 (0.41) AKR1B1ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102245587-A Trpv1 antagonists ABBOTT LAB 2011-11-16 CN disclosed
CN-102186836-A Trpv1 antagonists ABBOTT LAB 2011-09-14 CN disclosed