SCHEMBL27837726

SCHEMBL27837726

CC(=O)Oc1cc2cncnc2s1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
F2 P00734 1/20 0.34
GLA P06280 1/20 0.34
HPGD P15428 1/20 0.34
EGFR P00533 2/20 0.32
ALOX5 P09917 1/20 0.31
MAPT P10636 1/20 0.31
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16637562 0.85 HCAR2 (0.34)
SCHEMBL28818826 0.76 ALDH1A1 (0.33) ALDH1A1F2GLAHPGDEGFR
SCHEMBL27718543 0.74 CYP2A6 (0.53) ALDH1A1ALOX5
SCHEMBL6224494 0.73 POLB (0.42) ALDH1A1HPGDEGFRMAPT
SCHEMBL4800245 0.73 CSNK2A1 (0.46) ALDH1A1HPGDMAPT
SCHEMBL4908387 0.71 ALDH1A1 (0.42) ALDH1A1GLAMAPT
SCHEMBL29728017 0.71 ALDH1A1 (0.42) ALDH1A1GLAMAPT
SCHEMBL27586723 0.71 CYP2A6 (0.53) ALDH1A1GLAHPGDMAPTCA2
SCHEMBL5073476 0.70 DAPK3 (0.49)
SCHEMBL30396687 0.70 DAPK3 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104011054-A Thieno- and furo-pyrimidines and pyridines, useful as potassium channel inhibitors XENTION LTD 2014-08-27 CN disclosed
CN-102869669-A Heterocycloalkyl-containing thienopyrimidines for pharmaceutical compositions BOEHRINGER INGELHEIM INT 2013-01-09 CN disclosed
CN-102186857-A Thienopyrimidines for pharmaceutical compositions BOEHRINGER INGELHEIM INT 2011-09-14 CN disclosed