SCHEMBL27840909

SCHEMBL27840909

O=[N+]([O-])c1cccc(CSc2nccc(Cl)n2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.52
ALDH1A1 P00352 4/20 0.51
MAPT P10636 4/20 0.51
HTT P42858 3/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
HPGD P15428 1/20 0.51
LMNA P02545 2/20 0.50
POLB P06746 2/20 0.50
TSHR P16473 1/20 0.49
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C19 P33261 1/20 0.48
CDC7 O00311 1/20 0.48
DBF4 Q9UBU7 1/20 0.48
KDM4E B2RXH2 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
EGFR P00533 1/20 0.47
MET P08581 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6640173 0.81 CTSB (0.54) CTSBALDH1A1MAPTHTTL3MBTL1
SCHEMBL7509985 0.77 HSD17B10 (0.65) CTSBALDH1A1MAPTHTTL3MBTL1
SCHEMBL6638341 0.74 MAPK1 (0.47) ALDH1A1MAPTHTTL3MBTL1LMNA
SCHEMBL3244533 0.72 TSHR (0.65) CTSBALDH1A1MAPTHTTL3MBTL1
SCHEMBL3240297 0.72 TSHR (0.65) CTSBALDH1A1MAPTHTTL3MBTL1
SCHEMBL13722496 0.72 MEN1 (0.60) CTSBALDH1A1MAPTHTTL3MBTL1
SCHEMBL27682796 0.71 CYP1A2 (0.57) ALDH1A1MAPTHPGDLMNATSHR
SCHEMBL6637689 0.71 CTSB (0.54) CTSBALDH1A1MAPTHTTL3MBTL1
SCHEMBL5657175 0.70 MAPT (0.61) CTSBALDH1A1MAPTHTTLMNA
SCHEMBL10480613 0.70 MAPT (0.56) CTSBALDH1A1MAPTHTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102250097-A 6-alkyloxy-2-alkylthio-8-azapurine and synthesis thereof UNIV BEIJING CHEMICAL 2011-11-23 CN disclosed