SCHEMBL27846554

SCHEMBL27846554

Brc1ccc(/C(=C/c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.64
CYP19A1 P11511 5/20 0.57
CYP11B2 P19099 2/20 0.57
CYP1B1 Q16678 1/20 0.50
PTGS2 P35354 4/20 0.49
ESR2 Q92731 2/20 0.48
CYP2D6 P10635 1/20 0.47
KDM4E B2RXH2 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CTDSP1 Q9GZU7 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
AKR1C1 Q04828 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL987335 1.00 ESR1 (0.64) ESR1CYP19A1CYP11B2CYP1B1PTGS2
SCHEMBL14928213 1.00 ESR1 (0.64) ESR1CYP19A1CYP11B2CYP1B1PTGS2
SCHEMBL6517631 0.96 ESR1 (0.59) ESR1CYP19A1CYP11B2CYP1B1PTGS2
SCHEMBL6517636 0.96 ESR1 (0.59) ESR1CYP19A1CYP11B2CYP1B1PTGS2
SCHEMBL1652775 0.94 CYP19A1 (0.59) ESR1CYP19A1CYP11B2CYP1B1PTGS2
SCHEMBL6675573 0.90 ESR1 (0.53) ESR1CYP19A1CYP11B2CYP1B1PTGS2
SCHEMBL6675575 0.90 ESR1 (0.53) ESR1CYP19A1CYP11B2CYP1B1PTGS2
SCHEMBL4612465 0.89 ESR1 (0.78) ESR1CYP19A1CYP11B2PTGS2ESR2
SCHEMBL15607138 0.88 CYP19A1 (0.53) ESR1CYP19A1CYP11B2PTGS2ESR2
SCHEMBL21738730 0.87 ESR1 (0.62) ESR1CYP19A1CYP11B2PTGS2ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104341311-B Diamine compound and its preparation method and application 中山大学 2016-12-28 CN disclosed
CN-104341311-A Novel diamine compound, and preparation method and application thereof UNIV SUN YAT SEN 2015-02-11 CN disclosed
CN-102408342-B Fluorine-containing functional diamine monomer with large conjugated structure as well as synthesis method and application thereof UNIV SUN YAT SEN 2014-06-18 CN disclosed
CN-102766085-A Novel function diamine monomer containing carbazole and large conjugated structure and preparation method and application thereof UNIV SUN YAT SEN 2012-11-07 CN disclosed
CN-102408342-A Fluorine-containing functional diamine monomer with large conjugated structure as well as synthesis method and application thereof UNIV SUN YAT SEN 2012-04-11 CN disclosed