SCHEMBL27851069

SCHEMBL27851069

Nc1nc(NC(=O)O)cs1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.47
GABRA5 P31644 1/20 0.47
GABRB2 P47870 1/20 0.47
SMN1; SMN2 Q16637 4/20 0.43
NOS1 P29475 1/20 0.43
ALDH1A1 P00352 8/20 0.43
KDM4E B2RXH2 2/20 0.43
PIK3CG P48736 1/20 0.43
HTT P42858 1/20 0.42
MAPT P10636 5/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
NPC1 O15118 4/20 0.41
RAB9A P51151 2/20 0.41
LMNA P02545 3/20 0.40
CLK1 P49759 1/20 0.40
KDM6B O15054 1/20 0.39
KDM4A O75164 1/20 0.39
KDM4B O94953 1/20 0.39
KDM5C P41229 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10537469 0.85 GABRA5 (0.44) HSD17B10GABRA5GABRB2SMN1; SMN2NOS1
SCHEMBL2642609 0.82 PIK3CG (0.53) HSD17B10GABRA5GABRB2SMN1; SMN2NOS1
SCHEMBL2642900 0.78 HTT (0.47) HSD17B10GABRA5GABRB2SMN1; SMN2ALDH1A1
SCHEMBL16095753 0.78 GSTO1 (0.47) HSD17B10GABRA5GABRB2HTT
SCHEMBL21695368 0.78 GRM5 (0.45) SMN1; SMN2ALDH1A1KDM4EHTTMAPT
SCHEMBL4807003 0.76 HSD17B10 (0.51) HSD17B10GABRA5GABRB2SMN1; SMN2NOS1
SCHEMBL20558119 0.76 CDK5 (0.45) CCNA2CDK2CCNA1CDK5CDK5R1
SCHEMBL17675158 0.74 CA1 (0.41) SMN1; SMN2PIK3CGMEN1KMT2ACCNA2
SCHEMBL3138977 0.74 RXFP1 (0.57) SMN1; SMN2ALDH1A1KDM4EHTTMAPT
SCHEMBL20557462 0.73 CDK5 (0.43) MEN1KMT2ACCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101903378-B Aminotriazole derivatives ACTELION PHARMACEUTICALS LTD 2014-03-12 CN disclosed
CN-101903378-A Aminotriazole derivatives ACTELION PHARMACEUTICALS LTD 2010-12-01 CN disclosed