SCHEMBL27867342

SCHEMBL27867342

CNN1C(=O)c2c([N+](=O)[O-])cccc2C1(NC)NC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.41
S100A4 P26447 2/20 0.41
LMNA P02545 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
TSHR P16473 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
PTPRC P08575 1/20 0.38
KMT2A Q03164 3/20 0.37
MAPT P10636 1/20 0.37
RECQL P46063 1/20 0.37
MCL1 Q07820 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
ACHE P22303 1/20 0.35
GAA P10253 1/20 0.35
KDM4E B2RXH2 1/20 0.34
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2029915 0.72 S100A4 (0.46) TDP1S100A4LMNACA1CA2
SCHEMBL2030956 0.70 CA1 (0.48) TDP1S100A4LMNACA1CA2
SCHEMBL3039191 0.65 TDP1 (0.67) TDP1S100A4CA1CA2CA7
SCHEMBL1613571 0.63 S100A4 (0.46) TDP1S100A4LMNACA1CA2
SCHEMBL516272 0.62 LMNA (0.58) TDP1S100A4LMNACA1CA2
SCHEMBL30708932 0.62 LMNA (0.58) TDP1S100A4LMNACA1CA2
SCHEMBL472112 0.61 TDP1 (1.00) TDP1S100A4LMNATSHRSMN1; SMN2
SCHEMBL6051840 0.60 TSHR (0.69) TDP1S100A4LMNACA1CA2
SCHEMBL2524312 0.60 TDP1 (0.58) TDP1S100A4LMNATSHRSMN1; SMN2
SCHEMBL9397167 0.60 S100A4 (0.59) TDP1S100A4LMNACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102448955-B Aminopyrimidine Anticancer Compounds OSI PHARM INC 2014-06-18 CN disclosed
CN-102448955-A Aminopyrimidine Anticancer Compounds OSI PHARM INC 2012-05-09 CN disclosed