SCHEMBL27869722

SCHEMBL27869722

O=CC(CN1CCN(c2ccc3ccccc3n2)CC1)N1CC=C(c2cccc3ccsc23)CC1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.40
HRH3 Q9Y5N1 5/20 0.40
KDM4E B2RXH2 4/20 0.38
ALDH1A1 P00352 4/20 0.38
HTR3A P46098 3/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
CYP1A2 P05177 1/20 0.38
THPO P40225 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
RECQL P46063 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27886090 0.89 TSHR (0.30)
SCHEMBL27886019 0.88 DRD2 (0.32)
SCHEMBL27869721 0.88 HTR1A (0.40) HTR1AHRH3KDM4EALDH1A1HTR3A
SCHEMBL27886020 0.86 DRD4 (0.35) HTR1AALDH1A1
SCHEMBL27886124 0.81 KDM4E (0.48) HTR1AHRH3KDM4ELMNANPC1
SCHEMBL2179652 0.80 KDM4E (0.53) HTR1AHRH3KDM4EALDH1A1HTR3A
SCHEMBL27886089 0.75 PTGES (0.30)
SCHEMBL27886018 0.75 DRD2 (0.34) KDM4EALDH1A1LMNA
SCHEMBL27886017 0.73 DRD4 (0.39) HTR1AALDH1A1
SCHEMBL2195272 0.70 PDE10A (0.46) HTR1AKDM4EALDH1A1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102656162-A Novel (heterocycle/tetrahydropyridine)-(piperazinyl)-1-alcanone and (heterocycle/dihydropyrrolidine)-(piperazinyl)-1-alcanone derivatives, and use thereof as p75 inhibitors SANOFI SA 2012-09-05 CN claimed
CN-102656162-A Novel (heterocycle/tetrahydropyridine)-(piperazinyl)-1-alcanone and (heterocycle/dihydropyrrolidine)-(piperazinyl)-1-alcanone derivatives, and use thereof as p75 inhibitors SANOFI SA 2012-09-05 CN disclosed