SCHEMBL2787006

SCHEMBL2787006

O=C(NC1CCN(C(=O)O)C1)c1cncnc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 9/20 0.43
CTSL P07711 2/20 0.43
CTSB P07858 2/20 0.43
CTSK P43235 2/20 0.43
USP30 Q70CQ3 3/20 0.41
NPSR1 Q6W5P4 1/20 0.40
POLB P06746 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3217188 0.84 KDM5A (0.60) KDM5ACTSLCTSBCTSK
SCHEMBL5223407 0.83 KDM5A (0.57) KDM5ACTSLCTSBCTSKUSP30
SCHEMBL5223393 0.83 KDM5A (0.57) KDM5ACTSLCTSBCTSKUSP30
SCHEMBL994466 0.81 CTSL (0.63) KDM5ACTSLCTSBCTSKNPSR1
Bicarbonate SCHEMBL185416 0.78 ALDH1A1 (0.52) MEN1KMT2A
SCHEMBL185580 0.78 SMYD3 (0.54) MEN1KMT2A
SCHEMBL19133764 0.78 HDAC4 (0.47)
SCHEMBL25403939 0.77 CYP1A2 (0.57) KDM5ACTSLCTSBCTSKUSP30
SCHEMBL10212135 0.77 HDAC4 (0.52) DRD4
SCHEMBL25400740 0.77 CYP1A2 (0.57) KDM5ACTSLCTSBCTSKUSP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097374-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed