SCHEMBL27870698

SCHEMBL27870698

CCC(=O)OCC(C)(O)F

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.39
ALDH1A1 P00352 3/20 0.35
CYP1A2 P05177 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
BLM P54132 1/20 0.35
WRN Q14191 1/20 0.35
HIF1A Q16665 1/20 0.35
LMNA P02545 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HTT P42858 1/20 0.32
GAA P10253 2/20 0.32
MGAM O43451 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32
SOAT1 P35610 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
TRPA1 O75762 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27997782 0.84 ALDH1A1 (0.41) NAAAALDH1A1CYP1A2HPGDCYP2C19
SCHEMBL4450857 0.81 NAAA (0.41) NAAAALDH1A1CYP1A2HPGDCYP2C19
SCHEMBL974718 0.81 HTT (0.50) NAAAALDH1A1CYP1A2HPGDCYP2C19
SCHEMBL8402125 0.80 NAAA (0.38) NAAAALDH1A1CYP1A2HPGDCYP2C19
SCHEMBL12112110 0.80 NAAA (0.38) NAAAALDH1A1CYP1A2HPGDCYP2C19
Ammonia Solution, Strong SCHEMBL4621612 0.79 NAAA (0.40) NAAAALDH1A1CYP1A2HPGDCYP2C19
SCHEMBL28871728 0.78 NAAA (0.36) NAAAALDH1A1CYP1A2HPGDCYP2C19
SCHEMBL15281013 0.78 LMNA (0.45) NAAAALDH1A1CYP1A2HPGDCYP2C19
SCHEMBL14472846 0.78 NAAA (0.43) NAAAALDH1A1CYP1A2HPGDCYP2C19
SCHEMBL722286 0.78 NAAA (0.43) NAAAALDH1A1CYP1A2HPGDCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102471293-B Oxazine derivatives and their use as BACE inhibitors for the treatment of neurological disorders NOVARTIS AG (CH) 2014-10-01 CN disclosed
CN-102666507-B Oxazine derivatives and their use in the treatment of neurological disorders NOVARTIS AG 2014-09-17 CN disclosed
CN-103596569-A BACE-2 inhibitors for the treatment of metabolic disorders NOVARTIS AG 2014-02-19 CN disclosed
CN-103429588-A Crystalline oxazine derivative and its use as bace inhibitor NOVARTIS AG 2013-12-04 CN disclosed
CN-103429589-A Oxazine derivatives and their use in the treatment of neurological disorders NOVARTIS AG 2013-12-04 CN disclosed
CN-103403001-A Novel heterocyclic derivatives and their use in the treatment of neurological disorders NOVARTIS AG 2013-11-20 CN disclosed
CN-102666507-A Oxazine derivatives and their use in the treatment of neurological disorders NOVARTIS AG 2012-09-12 CN disclosed
CN-102471293-A Oxazine derivatives and their use as BACE inhibitors for the treatment of neurological disorders NOVARTIS AG 2012-05-23 CN disclosed