SCHEMBL27871237

SCHEMBL27871237

Nc1ccc(-c2ccc(NCCN3CCC(F)(F)CC3)nc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.45
ADRA1A P35348 3/20 0.45
DRD3 P35462 3/20 0.45
SIGMAR1 Q99720 3/20 0.45
ACHE P22303 1/20 0.42
HRH3 Q9Y5N1 2/20 0.41
KDR P35968 1/20 0.41
HRH4 Q9H3N8 1/20 0.41
ATR Q13535 1/20 0.41
MAP3K11 Q16584 1/20 0.40
FYN P06241 1/20 0.39
CRBN Q96SW2 1/20 0.39
MCHR1 Q99705 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
MAP4K4 O95819 1/20 0.38
SYK P43405 1/20 0.37
CD274 Q9NZQ7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1256889 0.99 DRD2 (0.44) DRD2ADRA1ADRD3SIGMAR1ACHE
SCHEMBL1256254 0.84 KDR (0.57) KDRATRFYNNPC1RAB9A
Hydrochloric Acid SCHEMBL1257055 0.82 KDR (0.56) KDRATRFYNNPC1RAB9A
SCHEMBL9958722 0.82 SIGMAR1 (0.45) DRD2ADRA1ADRD3SIGMAR1ACHE
SCHEMBL1257965 0.82 DRD2 (0.43) DRD2ADRA1ADRD3SIGMAR1ACHE
Acetic Acid SCHEMBL1256468 0.79 SIGMAR1 (0.43) DRD2ADRA1ADRD3SIGMAR1ACHE
SCHEMBL1255230 0.79 SIGMAR1 (0.48) SIGMAR1HRH3FYNNPC1RAB9A
SCHEMBL1256469 0.77 SIGMAR1 (0.41) DRD2ADRA1ADRD3SIGMAR1ACHE
SCHEMBL1257160 0.77 KDR (0.50) DRD2ADRA1ADRD3HRH3KDR
SCHEMBL1256232 0.76 CD274 (0.51) DRD2ADRA1ADRD3ACHEKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102470127-A Biaryl compounds and methods of use thereof AMBIT BIOSCIENCES CORP 2012-05-23 CN disclosed