SCHEMBL27878434

SCHEMBL27878434

COc1ccc(-c2ccc3[nH]c(C4CCN(OC(=O)C(C)(C)C)CC4)cc3c2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 15/20 0.46
TLR7 Q9NYK1 3/20 0.42
TLR8 Q9NR97 2/20 0.39
TLR9 Q9NR96 1/20 0.38
HTR2B P41595 1/20 0.37
PIK3CD O00329 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1980796 0.85 TLR7 (0.53) ABCB1TLR7TLR8PIK3CDPIK3CA
SCHEMBL27878458 0.81 HRH3 (0.42)
SCHEMBL1980058 0.77 TLR9 (0.54) ABCB1TLR7TLR8TLR9
SCHEMBL27862133 0.75 IDH1 (0.34) TLR7TLR8TLR9
Tert-Butyl Formate SCHEMBL27878435 0.75 TLR9 (0.45) ABCB1TLR7TLR8TLR9
SCHEMBL28309475 0.74 MEN1 (0.47)
SCHEMBL1981327 0.72 DPP4 (0.42) ABCB1TLR7TLR8TLR9HTR2B
SCHEMBL1981326 0.72 DPP4 (0.42) ABCB1TLR7TLR8TLR9HTR2B
SCHEMBL1980557 0.72 CTSS (0.41) ABCB1TLR7TLR8TLR9
SCHEMBL1980560 0.72 CTSS (0.41) ABCB1TLR7TLR8TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102753524-B Bicyclic derivatives useful as inhibitors of dpp-1 ANSSEN PHARMACEUTICA NV 2014-11-05 CN disclosed
CN-102753524-A Bicyclic derivatives useful as inhibitors of dpp-1 ANSSEN PHARMACEUTICA NV 2012-10-24 CN disclosed