SCHEMBL27890843

SCHEMBL27890843

Nc1ccc(Cc2c[nH]c3nccc(-c4ccccc4)c23)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 4/20 0.47
MET P08581 1/20 0.41
ROCK1 Q13464 4/20 0.40
ROCK2 O75116 3/20 0.40
CDC42BPB Q9Y5S2 1/20 0.40
GSK3B P49841 3/20 0.39
JAK2 O60674 4/20 0.38
CHUK O15111 3/20 0.38
PRKD3 O94806 3/20 0.38
MAP4K4 O95819 3/20 0.38
FGFR1 P11362 3/20 0.38
PRKACA P17612 3/20 0.38
KDR P35968 3/20 0.38
CLK2 P49760 3/20 0.38
CDK5 Q00535 3/20 0.38
MAP4K2 Q12851 3/20 0.38
PRKAA1 Q13131 3/20 0.38
DYRK1A Q13627 3/20 0.38
AURKB Q96GD4 3/20 0.38
ALK Q9UM73 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL857300 0.86 LRRK2 (0.47) LRRK2METROCK1JAK2CHUK
SCHEMBL1887197 0.77 ROCK2 (0.36) LRRK2METROCK1ROCK2CDC42BPB
SCHEMBL3813831 0.75 MET (0.65) METROCK1ROCK2GSK3BPRKD3
SCHEMBL1888240 0.72 CYP3A4 (0.49) KDRAURKBCSF1RNTRK3FLT1
SCHEMBL26953278 0.72 SGK1 (0.57) LRRK2ROCK1ROCK2GSK3BJAK2
SCHEMBL31735012 0.72 SGK1 (0.57) LRRK2ROCK1ROCK2GSK3BJAK2
SCHEMBL857282 0.70 LRRK2 (0.51) LRRK2GSK3BCDK5CDK8CDK9
SCHEMBL20086205 0.70 LRRK2 (0.50) LRRK2GSK3BCDK5DYRK1ACDK8
SCHEMBL857855 0.68 SIK1 (0.51) LRRK2CSF1RCDK8FYNMAPK1
SCHEMBL22988837 0.68 MET (0.41) METFGFR1KDRAURKBCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102695417-A Compounds and methods for kinase modulation and indications therefor PLEXXIKON INC 2012-09-26 CN disclosed