SCHEMBL27891776

SCHEMBL27891776

COCc1nc(C(=O)OCc2ccccc2)c(Oc2ccccc2)c2ccc(Oc3ccccc3)cc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 3/20 0.44
TOP2B Q02880 3/20 0.44
THRA P10827 8/20 0.42
THRB P10828 8/20 0.42
EGLN1 Q9GZT9 6/20 0.42
EGLN2 Q96KS0 3/20 0.42
MMP1 P03956 2/20 0.40
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
GABRA1 P14867 1/20 0.40
HPGD P15428 1/20 0.40
GABRB1 P18505 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40
GABRA2 P47869 1/20 0.40
GABRB2 P47870 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL522420 0.94 GABRA1 (0.42) TOP2ATOP2BTHRATHRBEGLN1
SCHEMBL522570 0.84 MCL1 (0.46) THRATHRBEGLN1BBOX1SLC6A2
SCHEMBL523582 0.80 THRA (0.49) THRATHRBEGLN1EGLN2BBOX1
SCHEMBL523190 0.80 EGLN1 (0.51) TOP2ATOP2BTHRATHRBEGLN1
SCHEMBL523555 0.79 ALDH1A1 (0.46) GABRPGABRDALDH1A1MAPTGABRA1
SCHEMBL522588 0.78 EGLN1 (0.53) TOP2ATOP2BTHRATHRBEGLN1
SCHEMBL523204 0.77 MCL1 (0.41) TOP2ATOP2BTHRATHRBEGLN1
SCHEMBL15433916 0.76 THRA (0.43) THRATHRBEGLN1EGLN2BBOX1
SCHEMBL28488469 0.75 EGLN1 (0.64) THRATHRBEGLN1EGLN2BBOX1
SCHEMBL522739 0.75 POLB (0.48) EGLN1EGLN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102718708-A Novel nitrogen-containing heteroaryl compounds and methods of use thereof FIBROGEN INC 2012-10-10 CN disclosed