Isoxazole

Isoxazole

SCHEMBL27896201

c1cnoc1.c1coc(-c2ncco2)c1

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.45
NPC1 O15118 10/20 0.39
RAB9A P51151 10/20 0.39
HSD17B10 Q99714 10/20 0.39
SMN1; SMN2 Q16637 6/20 0.39
TP53 P04637 5/20 0.39
POLB P06746 4/20 0.39
PKM P14618 3/20 0.39
ALDH1A1 P00352 11/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
KDM4E B2RXH2 10/20 0.38
HPGD P15428 8/20 0.38
MAPT P10636 7/20 0.38
ALOX15 P16050 2/20 0.38
CASP1 P29466 2/20 0.38
PTPN7 P35236 2/20 0.38
RECQL P46063 2/20 0.38
BLM P54132 2/20 0.38
CASP7 P55210 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3980455 0.87 ALDH1A1 (0.48) NPC1RAB9AHSD17B10SMN1; SMN2TP53
Isoxazole SCHEMBL27894024 0.72 RAB9A (0.41) PARP1NPC1RAB9AHSD17B10SMN1; SMN2
SCHEMBL28928829 0.71 BRD4 (0.43) NPC1RAB9AHSD17B10SMN1; SMN2TP53
SCHEMBL3263841 0.71 RAB9A (0.63) NPC1RAB9AHSD17B10SMN1; SMN2TP53
Isoxazole SCHEMBL28776356 0.70 MEN1 (0.44) PARP1ALDH1A1MEN1KMT2AHPGDS
Isoxazole SCHEMBL28638568 0.68 PARP1 (0.54) PARP1
Isoxazole SCHEMBL2679369 0.67 PARP1 (1.00) PARP1
Isoxazole SCHEMBL1318 0.67
Isoxazole SCHEMBL393230 0.67
SCHEMBL19528998 0.66 NOTUM (0.41) NPC1RAB9AHSD17B10SMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102762208-A Pyrazolopyrimidines and related heterocycles as ck2 inhibitors CYLENE PHARMACEUTICALS INC 2012-10-31 CN disclosed